SCHEMBL15564166

SCHEMBL15564166

Cc1cccc(CCn2nc(O)c(=O)[nH]c2=O)c1

nearest known ligand 0.57

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DAO P14920 8/20 0.57
GPR84 Q9NQS5 1/20 0.46
HRH3 Q9Y5N1 1/20 0.43
ALDH1A1 P00352 1/20 0.40
TSHR P16473 1/20 0.40
KDM1A O60341 1/20 0.40
IDO1 P14902 1/20 0.40
XIAP P98170 1/20 0.39
TAAR1 Q96RJ0 1/20 0.39
MEN1 O00255 1/20 0.39
TP53 P04637 1/20 0.39
HTT P42858 1/20 0.39
KMT2A Q03164 1/20 0.39
HSD17B10 Q99714 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15564228 0.93 DAO (0.51) DAOGPR84HRH3ALDH1A1TSHR
SCHEMBL15564534 0.87 DAO (0.60) DAOTAAR1
SCHEMBL15564020 0.87 DAO (0.60) DAOTAAR1
SCHEMBL15564255 0.85 DAO (0.57) DAO
SCHEMBL16968231 0.85 DAO (0.57) DAOGPR84HRH3ALDH1A1TSHR
SCHEMBL15564061 0.84 DAO (0.60) DAOHRH3TAAR1
SCHEMBL15563972 0.84 DAO (0.54) DAOGPR84HRH3ALDH1A1
SCHEMBL15564271 0.84 DAO (0.55) DAOALDH1A1HTTKMT2A
SCHEMBL15563813 0.81 DAO (0.60) DAOTAAR1KMT2A
SCHEMBL15564151 0.81 DAO (0.61) DAOMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9505753-B2 Inhibitors of D-amino acid oxidase THE JOHNS HOPKINS UNIVERSITY (US) 2016-11-29 US claimed
US-20150218156-A1 INHIBITORS OF D-AMINO ACID OXIDASE THE JOHNS HOPKINS UNIVERSITY (US) 2015-08-06 US claimed
WO-2014025993-A1 INHIBITORS OF D-AMINO ACID OXIDASE THE JOHNS HOPKINS UNIVERSITY (US) 2014-02-13 WO claimed
US-9505753-B2 Inhibitors of D-amino acid oxidase THE JOHNS HOPKINS UNIVERSITY (US) 2016-11-29 US disclosed
US-20150218156-A1 INHIBITORS OF D-AMINO ACID OXIDASE THE JOHNS HOPKINS UNIVERSITY (US) 2015-08-06 US disclosed
WO-2014025993-A1 INHIBITORS OF D-AMINO ACID OXIDASE THE JOHNS HOPKINS UNIVERSITY (US) 2014-02-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150218156-A1 INHIBITORS OF D-AMINO ACID OXIDASE DDO, DAO, GRIN2A DAO 2/4885GPR84 273/4885HRH3 1538/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.