SCHEMBL15569333

SCHEMBL15569333

CC1CCC(C(C)C)C(CC(=O)NC2CC2)C1

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 4/20 0.48
TRPM8 Q7Z2W7 4/20 0.43
TRPA1 O75762 2/20 0.43
TRPV1 Q8NER1 5/20 0.41
MEN1 O00255 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3793761 0.84 EPHX1 (0.47) EPHX1TRPM8TRPA1TRPV1
SCHEMBL694600 0.81 EPHX1 (0.49) EPHX1TRPM8TRPA1TRPV1
SCHEMBL9951281 0.80 EPHX1 (0.44) EPHX1TRPM8TRPA1TRPV1
SCHEMBL19719724 0.80 EPHX1 (0.44) EPHX1TRPM8TRPA1TRPV1
SCHEMBL24168644 0.80 EPHX1 (0.44) EPHX1TRPM8TRPA1TRPV1
SCHEMBL694116 0.79 EPHX1 (0.43) EPHX1TRPM8TRPA1TRPV1
SCHEMBL29090851 0.79 EPHX1 (0.43) EPHX1TRPM8TRPA1TRPV1
SCHEMBL29152577 0.79 EPHX1 (0.46) EPHX1TRPM8TRPA1TRPV1
SCHEMBL9951688 0.78 EPHX1 (0.51) EPHX1TRPM8TRPA1TRPV1
SCHEMBL9951381 0.78 EPHX1 (0.51) EPHX1TRPM8TRPA1TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4247791-A2 NEW COOLANTS, AND PREPARATIONS CONTAINING SAME Symrise AG (DE) 2023-09-27 EP claimed
WO-2023143741-A1 NEW COOLANTS, AND PREPARATIONS CONTAINING SAME SYMRISE AG (DE) 2023-08-03 WO claimed
WO-2023117119-A1 ACTIVE INGREDIENTS WITH SIALAGOGUE AND TINGLING/FIZZY EFFECT, AND PREPARATIONS CONTAINING SAME SYMRISE AG (DE) 2023-06-29 WO claimed
WO-2022105986-A1 NOVEL COOLING AGENTS AND PREPARATIONS CONTAINING SAME SYMRISE AG (DE) 2022-05-27 WO claimed
WO-2022106452-A2 NEW COOLANTS, AND PREPARATIONS CONTAINING SAME SYMRISE AG (DE) 2022-05-27 WO claimed
WO-2023144326-A1 NEW COOLANTS, AND PREPARATIONS CONTAINING SAME SYMRISE AG (DE) 2023-08-03 WO disclosed
WO-2023092212-A1 FLAVOURING AGENT, COMPOSITION, PRODUCTION METHOD AND USE OF AROMATISING AND FLAVOURING AGENTS BASED ON VANILLA EXTRACTS UNIVERSIDADE FEDERAL DO ESTADO DO RIO DE JANEIRO (BR) 2023-06-01 WO disclosed
EP-2884958-B1 COSMETIC COMPOUNDS HAVING TIME-DELAYED ACTIVE INGREDIENT RELEASE HENKEL AG & CO KGAA (DE) 2017-03-29 EP disclosed
US-9517195-B2 Cosmetic compounds having time-delayed active ingredient release HENKEL AG & CO. KGAA (DE) 2016-12-13 US disclosed
EP-2884958-A2 COSMETIC COMPOUNDS HAVING TIME-DELAYED ACTIVE INGREDIENT RELEASE Henkel AG&Co. KGAA (DE) 2015-06-24 EP disclosed
US-20150157552-A1 COSMETIC COMPOUNDS HAVING TIME-DELAYED ACTIVE INGREDIENT RELEASE HENKEL AG & CO. KGAA (DE) 2015-06-11 US disclosed
WO-2014198366-A1 GLOVE WITH A COOLING EFFECT CARL FREUDENBERG KG (DE) 2014-12-18 WO disclosed
WO-2014026842-A2 COSMETIC COMPOUNDS HAVING TIME-DELAYED ACTIVE INGREDIENT RELEASE HENKEL AG & CO. KGAA (DE) 2014-02-20 WO disclosed