SCHEMBL15570495

SCHEMBL15570495

O=C(O)c1cnc2c(Br)n[nH]c2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 4/20 0.41
POLB P06746 1/20 0.41
DYRK1A Q13627 1/20 0.40
PSMD14 O00487 1/20 0.39
DYRK1B Q9Y463 1/20 0.37
MGAM O43451 1/20 0.37
KDM4E B2RXH2 2/20 0.36
KDM4A O75164 1/20 0.36
KDM5C P41229 1/20 0.36
KDM4C Q9H3R0 1/20 0.36
KDM2A Q9Y2K7 1/20 0.36
KDM3A Q9Y4C1 1/20 0.36
P4HA1 P13674 3/20 0.35
P4HTM Q9NXG6 2/20 0.35
MIF P14174 1/20 0.34
MAP2K4 P45985 5/20 0.34
MAPK1 P28482 3/20 0.34
MAPK6 Q16659 3/20 0.34
MAPKAPK3 Q16644 2/20 0.34
GABRP O00591 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13552110 0.80 HCAR2 (0.44) HCAR2POLBPSMD14MGAMKDM4E
SCHEMBL28586933 0.73 HCAR2 (0.41) HCAR2POLBDYRK1BMGAMKDM4E
SCHEMBL13386987 0.73 HCAR2 (0.41) HCAR2POLBPSMD14MGAMKDM4E
Hydrochloric Acid SCHEMBL13386995 0.72 HCAR2 (0.40) HCAR2POLBPSMD14MGAMKDM4E
SCHEMBL30967983 0.72 DYRK1A (0.44) DYRK1APSMD14KDM4E
SCHEMBL9818232 0.71 MAP2K4 (0.50) DYRK1ADYRK1BKDM4EMAP2K4MAPK1
SCHEMBL31523324 0.71 MAP2K4 (0.50) DYRK1ADYRK1BKDM4EMAP2K4MAPK1
SCHEMBL30792836 0.69 HCAR2 (0.50) HCAR2POLBPSMD14MGAMKDM4E
SCHEMBL487368 0.69 HCAR2 (0.50) HCAR2POLBPSMD14MGAMKDM4E
SCHEMBL1759261 0.67 DYRK1A (0.52) HCAR2POLBDYRK1AMGAMKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2884981-A2 4-HETEROARYL SUBSTITUTED BENZOIC ACID COMPOUNDS AS RORgammaT INHIBITORS AND USES THEREOF Merck Sharp & Dohme Corp. (US) 2015-06-24 EP disclosed
WO-2014028589-A2 4-HETEROARYL SUBSTITUTED BENZOIC ACID COMPOUNDS AS RORgammaT INHIBITORS AND USES THEREOF MERCK SHARP & DOHME CORP. (US) 2014-02-20 WO disclosed