SCHEMBL15580681

SCHEMBL15580681

C[C@H](c1ccc(Oc2nc(C(F)(F)F)ccc2C(=O)O)cc1Cl)[C@@](O)(c1ccc2[nH]c(=O)n(C)c2c1)C(F)(F)F

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.33
PDE2A O00408 3/20 0.31
CDK2 P24941 1/20 0.31
AKT1 P31749 1/20 0.31
BRD4 O60885 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL474430 0.88 CMA1 (0.34) BRD4
SCHEMBL12164077 0.88 CMA1 (0.34) BRD4
SCHEMBL474551 0.76 BRD4 (0.38) BRD4
SCHEMBL12164033 0.76 BRD4 (0.38) BRD4
SCHEMBL474403 0.75 PTGER4 (0.41)
SCHEMBL12164066 0.75 BRD4 (0.36) BRD4
SCHEMBL12164064 0.75 PTGER4 (0.41)
SCHEMBL474361 0.75 BRD4 (0.36) BRD4
SCHEMBL474429 0.75 CMA1 (0.34) BRD4
SCHEMBL12164091 0.75 CMA1 (0.34) BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-B1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS HOFFMANN LA ROCHE (CH) 2014-03-19 EP disclosed