SCHEMBL15613640

SCHEMBL15613640

COc1ccc(COc2cccc(Oc3ccc(-c4nn(C5CCCC5)c5ncnc(N)c45)cc3)c2)cc1

nearest known ligand 0.69

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BTK Q06187 12/20 0.69
LCK P06239 2/20 0.69
LYN P07948 1/20 0.69
NUDT14 O95848 1/20 0.60
NUDT5 Q9UKK9 1/20 0.60
EGFR P00533 11/20 0.58
SRC P12931 7/20 0.58
KDR P35968 7/20 0.58
PIK3CD O00329 7/20 0.58
PIK3CA P42336 7/20 0.58
PIK3CB P42338 7/20 0.58
PIK3CG P48736 7/20 0.58
PRKDC P78527 7/20 0.58
ABL1 P00519 6/20 0.58
HCK P08631 6/20 0.58
MTOR P42345 6/20 0.58
EPHB4 P54760 6/20 0.58
PI4KB Q9UBF8 6/20 0.58
TEK Q02763 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15613639 0.94 BTK (0.68) BTKLCKLYNNUDT14NUDT5
SCHEMBL16886143 0.93 BTK (0.69) BTKLCKLYNNUDT14NUDT5
SCHEMBL15613546 0.92 BTK (0.79) BTKLCKLYNNUDT14NUDT5
SCHEMBL15613472 0.92 BTK (0.69) BTKLCKLYNNUDT14NUDT5
SCHEMBL6431315 0.91 BTK (0.80) BTKLCKLYNNUDT14NUDT5
SCHEMBL15613695 0.87 BTK (0.79) BTKLCKLYNNUDT14NUDT5
SCHEMBL16886154 0.86 BTK (0.71) BTKLCKLYNNUDT14NUDT5
SCHEMBL15613699 0.85 BTK (0.67) BTKLCKLYNNUDT14NUDT5
SCHEMBL16886144 0.84 BTK (0.68) BTKLCKLYNNUDT14NUDT5
SCHEMBL15613469 0.84 BTK (0.65) BTKLCKLYNNUDT14NUDT5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9796716-B2 Selective inhibitors of Tec and Src protein kinase families PHARMASCIENCE, INC. (CA) 2017-10-24 US disclosed
US-9796716-B2 Selective inhibitors of Tec and Src protein kinase families PHARMASCIENCE, INC. (CA) 2017-10-24 US disclosed
US-20150191473-A1 PROTEIN KINASE INHIBITORS PHARMASCIENCE, INC. (CA) 2015-07-09 US disclosed
US-20150191473-A1 PROTEIN KINASE INHIBITORS PHARMASCIENCE, INC. (CA) 2015-07-09 US disclosed
WO-2013177668-A1 PROTEIN KINASE INHIBITORS PHARMASCIENCE, INC. (CA) 2013-12-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150191473-A1 PROTEIN KINASE INHIBITORS TEC, SRC, LCK BTK 10/4885LCK 3/4885LYN 30/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.