SCHEMBL15640367

SCHEMBL15640367

Cn1c(-c2ccccc2)cc2cc(S(=O)(=O)NC3CCC(C(=O)NC(CC(=O)O)c4ccccc4)CC3)ccc21

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGDR Q13258 1/20 0.42
ITGB3 P05106 3/20 0.42
ITGAV P06756 1/20 0.42
POLB P06746 2/20 0.40
TYK2 P29597 1/20 0.40
ITGA2B P08514 2/20 0.39
CASP3 P42574 1/20 0.39
F11 P03951 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CCR5 P51681 1/20 0.38
NR1H2 P55055 1/20 0.38
ITGB1 P05556 1/20 0.37
ITGA4 P13612 1/20 0.37
MTNR1A P48039 1/20 0.37
MTNR1B P49286 1/20 0.37
IDH2 P48735 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15640366 1.00 PTGDR (0.42) PTGDRITGB3ITGAVPOLBTYK2
SCHEMBL15640365 1.00 PTGDR (0.42) PTGDRITGB3ITGAVPOLBTYK2
SCHEMBL517705 0.90 NR1H2 (0.44) NR1H2
SCHEMBL517704 0.90 NR1H2 (0.44) NR1H2
SCHEMBL15640282 0.87 PTGDR (0.48) PTGDRPOLBTYK2CCR5NR1H2
SCHEMBL15640283 0.87 PTGDR (0.48) PTGDRPOLBTYK2CCR5NR1H2
SCHEMBL517056 0.85 NR1H2 (0.41) PTGDRPOLBTYK2NR1H2MTNR1A
SCHEMBL517055 0.85 NR1H2 (0.41) PTGDRPOLBTYK2NR1H2MTNR1A
SCHEMBL15640459 0.85 PTGDR (0.46) PTGDRPOLBTYK2CCR5NR1H2
SCHEMBL15640458 0.85 PTGDR (0.46) PTGDRPOLBTYK2CCR5NR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2598486-B1 BICYCLIC ACETYL-COA CARBOXYLASE INHIBITORS NOVARTIS AG (CH) 2017-06-28 EP claimed
US-8697739-B2 Bicyclic acetyl-CoA carboxylase inhibitors and uses thereof NOVARTIS AG (CH) 2014-04-15 US claimed
EP-2598486-B1 BICYCLIC ACETYL-COA CARBOXYLASE INHIBITORS NOVARTIS AG (CH) 2017-06-28 EP disclosed