SCHEMBL15664448

SCHEMBL15664448

COc1cc2c(Oc3ccc(Nc4nnc(-c5ccccc5)c5ccccc45)cc3)ccnc2cc1OCc1ccccc1

nearest known ligand 0.63

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
FGFR2 P21802 5/20 0.63
PDGFRA P16234 3/20 0.52
KDR P35968 3/20 0.52
MET P08581 3/20 0.50
KIT P10721 2/20 0.50
EGFR P00533 2/20 0.50
RIPK2 O43353 1/20 0.50
EPHB2 P29323 1/20 0.50
RET P07949 2/20 0.49
AXL P30530 1/20 0.49
LMNA P02545 1/20 0.48
MAPT P10636 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2207029 0.93 FGFR2 (0.72) FGFR2PDGFRAKDRKITEGFR
SCHEMBL2207343 0.90 FGFR2 (0.63) FGFR2PDGFRAKDRMETKIT
SCHEMBL2208900 0.87 FGFR2 (0.63) FGFR2PDGFRAKDRKITAXL
SCHEMBL14047121 0.86 FGFR2 (0.62) FGFR2PDGFRAKDRKITRET
SCHEMBL2208407 0.84 FGFR2 (0.71) FGFR2PDGFRAKDRKIT
SCHEMBL2210992 0.84 FGFR2 (0.58) FGFR2KDREGFRLMNAMAPT
SCHEMBL2211767 0.84 FGFR2 (0.58) FGFR2KDREGFRLMNAMAPT
SCHEMBL2210071 0.84 FGFR2 (0.59) FGFR2PDGFRAKDRMETKIT
SCHEMBL2210388 0.83 FGFR2 (0.63) FGFR2PDGFRAKDRKITAXL
SCHEMBL4486596 0.82 FGFR2 (0.81) FGFR2PDGFRAKDRMETKIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2137177-B1 AURORA KINASE MODULATORS AND METHOD OF USE AMGEN INC (US) 2014-05-07 EP disclosed