SCHEMBL15711490

SCHEMBL15711490

Cc1ccc(N/N=C\C=N)c(C(=O)N2CC(c3nc4cc(Cl)cnc4o3)CC[C@H]2C)c1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 18/20 0.36
HCRTR1 O43613 8/20 0.36
NR1I2 O75469 1/20 0.36
ADRA2B P18089 1/20 0.36
KCNH2 Q12809 1/20 0.36
KDM4E B2RXH2 1/20 0.34
NPC1 O15118 1/20 0.34
ALDH1A1 P00352 1/20 0.34
TP53 P04637 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
HPGD P15428 1/20 0.34
CYP2C19 P33261 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HSD17B10 Q99714 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15944028 1.00 HCRTR2 (0.36) HCRTR2HCRTR1NR1I2ADRA2BKCNH2
SCHEMBL15944065 0.88 HCRTR1 (0.47) HCRTR2HCRTR1NR1I2ADRA2BKCNH2
SCHEMBL15711500 0.88 HCRTR2 (0.41) HCRTR2HCRTR1
SCHEMBL15943988 0.88 HCRTR2 (0.41) HCRTR2HCRTR1
SCHEMBL15944014 0.82 HCRTR2 (0.42) HCRTR2HCRTR1NR1I2ADRA2BKCNH2
SCHEMBL15711496 0.82 HCRTR2 (0.42) HCRTR2HCRTR1NR1I2ADRA2BKCNH2
SCHEMBL15711482 0.80 HCRTR2 (0.40) HCRTR2HCRTR1NR1I2ADRA2BKCNH2
SCHEMBL15673220 0.79 HCRTR2 (0.55) HCRTR2HCRTR1NR1I2ADRA2BKCNH2
SCHEMBL15944012 0.79 HCRTR2 (0.43) HCRTR2HCRTR1NR1I2ADRA2BKCNH2
SCHEMBL15944064 0.78 HCRTR2 (0.41) HCRTR2HCRTR1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2730573-A1 METHYLPIPERIDINE DERIVATIVE Taisho Pharmaceutical Co., Ltd. (JP) 2014-05-14 EP disclosed