SCHEMBL15719941

SCHEMBL15719941

Nc1ncc(S)c(-c2ccccc2)n1

nearest known ligand 0.57

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 16/20 0.57
ADORA2A P29274 12/20 0.57
LMNA P02545 1/20 0.53
NUDT1 P36639 1/20 0.47
GFER P55789 1/20 0.46
KMT2A Q03164 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14127720 0.80 ADORA1 (0.61) ADORA1ADORA2ALMNANUDT1GFER
SCHEMBL4582424 0.78 ADORA1 (0.83) ADORA1ADORA2AGFERKMT2A
SCHEMBL6980294 0.77 KDM4E (0.52) ADORA1ADORA2ALMNAKMT2A
SCHEMBL27324019 0.77 MAPT (0.54) LMNA
SCHEMBL24309649 0.77 ADORA1 (0.63) ADORA1ADORA2ALMNANUDT1
SCHEMBL13377688 0.77 ADORA1 (0.57) ADORA1ADORA2ALMNANUDT1GFER
SCHEMBL7147862 0.77 ADORA1 (0.57) ADORA1ADORA2ALMNANUDT1
SCHEMBL508845 0.77 ADORA1 (0.57) ADORA1ADORA2ALMNANUDT1
Ammonia Solution, Strong SCHEMBL28877790 0.77 ADORA1 (0.81) ADORA1ADORA2AGFERKMT2A
SCHEMBL3021383 0.77 ADORA1 (0.59) ADORA1ADORA2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2920153-A1 4-(ORTHO)-FLUOROPHENYL-5-FLUOROPYRIMIDIN-2-YL AMINES CONTAINING A SULFOXIMINE GROUP Bayer Pharma Aktiengesellschaft (DE) 2015-09-23 EP disclosed
WO-2014076028-A1 4-(ORTHO)-FLUOROPHENYL-5-FLUOROPYRIMIDIN-2-YL AMINES CONTAINING A SULFOXIMINE GROUP BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2014-05-22 WO disclosed