SCHEMBL15768106

SCHEMBL15768106

CN(C)C(=O)c1cnn(C)c1C(=O)Nc1ccn2cc(-c3c[c]ccc3)nc2n1

nearest known ligand 0.68

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 20/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6916062 0.89 PDE10A (0.83) PDE10A
SCHEMBL15768108 0.86 PDE10A (0.59) PDE10A
SCHEMBL2385774 0.85 PDE10A (0.69) PDE10A
SCHEMBL2384173 0.85 PDE10A (0.68) PDE10A
SCHEMBL12316451 0.84 PDE10A (0.67) PDE10A
SCHEMBL2401366 0.82 PDE10A (0.64) PDE10A
SCHEMBL2373731 0.81 PDE10A (1.00) PDE10A
SCHEMBL6915732 0.81 PDE10A (0.78) PDE10A
SCHEMBL2395207 0.81 PDE10A (0.65) PDE10A
SCHEMBL12266628 0.80 PDE10A (0.85) PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2552918-B1 N-(IMIDAZOPYRIMIDIN-7-YL)-HETEROARYLAMIDE DERIVATIVES AND THEIR USE AS PDE10A INHIBITORS HOFFMANN LA ROCHE (CH) 2014-06-11 EP claimed