Quinapril

Quinapril

SCHEMBL15813

CCOC(=O)[C@H](CCc1ccccc1)N[C@@H](C)C(=O)N1Cc2ccccc2C[C@H]1C(=O)O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACE

The experimentally established mechanism targets of Quinapril. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ACE known ✓ P12821 16/20 1.00
ABCB11 O95342 2/20 1.00
PDE3A Q14432 1/20 0.80
LMNA P02545 1/20 0.70
SMN1; SMN2 Q16637 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Quinapril SCHEMBL13575806 1.00 ACE (1.00) ACEABCB11PDE3ALMNASMN1; SMN2
Quinapril SCHEMBL29380303 1.00 ACE (1.00) ACEABCB11PDE3ALMNASMN1; SMN2
Quinapril SCHEMBL29846170 1.00 ACE (1.00) ACEABCB11PDE3ALMNASMN1; SMN2
Quinapril SCHEMBL678447 1.00 ACE (1.00) ACEABCB11PDE3ALMNASMN1; SMN2
Quinapril SCHEMBL11286555 1.00 ACE (1.00) ACEABCB11PDE3ALMNASMN1; SMN2
Quinapril SCHEMBL11294979 1.00 ACE (1.00) ACEABCB11PDE3ALMNASMN1; SMN2
Quinapril SCHEMBL19361887 1.00 ACE (1.00) ACEABCB11PDE3ALMNASMN1; SMN2
Quinapril SCHEMBL994608 1.00 ACE (1.00) ACEABCB11PDE3ALMNASMN1; SMN2
Quinapril SCHEMBL9094436 1.00 ACE (1.00) ACEABCB11PDE3ALMNASMN1; SMN2
Quinapril SCHEMBL11286551 1.00 ACE (1.00) ACEABCB11PDE3ALMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 34108 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3607938-B1 PHARMACEUTICAL COMPOSITION SOVIC BRKICIC LJILJANA (HR) 2026-05-27 EP claimed
WO-2026087680-A1 TREATMENT FOR CARDIOVASCULAR DISEASE SAPREME TECHNOLOGIES B.V. (NL) 2026-04-30 WO claimed
EP-4731194-A1 MATERIALS AND METHODS FOR MITIGATING THE PRESENCE OF NITROSAMINES IN PACKAGING USING AN ACTIVE AGENT CSP Technologies, Inc. (US) 2026-04-29 EP claimed
US-12605345-B2 Transdermal drug delivery system BioPhysics Pharma, Inc. (US) 2026-04-21 US claimed
US-20260083968-A1 COMPOSITIONS, SYSTEMS, AND METHODS FOR TREATING CANCER USING TUMOR TREATING FIELDS (TTFIELDS) AND ACE INHIBITORS NOVOCURE GMBH (CH) 2026-03-26 US claimed
EP-4710928-A2 METHODS OF TREATING IGA NEPHROPATHY WITH ATRASENTAN Chinook Therapeutics, Inc. (US) 2026-03-18 EP claimed
EP-4691556-A2 HUMANIZED ANTI-ACTH ANTIBODIES AND USE THEREOF H. Lundbeck A/S (DK) 2026-02-11 EP claimed
EP-4687805-A1 MATERIALS AND METHODS FOR MITIGATING THE PRESENCE OF NITROSAMINES IN PACKAGING USING ACTIVATED CARBON OR A DERIVATIVE THEREOF CSP Technologies, Inc. (US) 2026-02-11 EP claimed
US-20260027008-A1 MATERIALS AND METHODS FOR MITIGATING THE PRESENCE OF NITROSAMINES IN PACKAGING USING ACTIVATED CARBON OR A DERIVATIVE THEREOF CSP TECHNOLOGIES, INC. 2026-01-29 US claimed
EP-4684832-A2 POTASSIUM-BINDING AGENTS FOR TREATING HYPERTENSION AND HYPERKALEMIA Vifor (International) Ltd. (CH) 2026-01-28 EP claimed
US-4793998-A ASCORBIC ACID AS STABILIZER FOR ANGIOTENSIN CONVERTING ENZYME WARNER-LAMBERT COMPANY (US) 1988-12-27 US claimed
EP-0285992-A1 Crystalline quinapril and a process for producing the same WARNER-LAMBERT COMPANY (US) 1988-10-12 EP claimed
EP-0280999-A2 Stabilized pharmaceutical compositions containing angiotensin-converting enzyme inhibitors WARNER-LAMBERT COMPANY (US) 1988-09-07 EP claimed
EP-0135182-B1 PROCESS FOR THE PRODUCTION OF N-ALKYLATED DIPEPTIDES AND OF THEIR ESTERS HOECHST AKTIENGESELLSCHAFT (DE) 1988-07-27 EP claimed
US-4743450-A ANGIOTENSION CONVERTING ENZYME INHIBITORS WARNER-LAMBERT COMPANY (US) 1988-05-10 US claimed
EP-0265685-A2 Combination of ACE inhibitors with calcium antagonists, and their use in medicines HOECHST AKTIENGESELLSCHAFT (DE) 1988-05-04 EP claimed
EP-0264887-A1 Drug compositions stabilized against oxidation and discoloration WARNER-LAMBERT COMPANY (US) 1988-04-27 EP claimed
EP-0264888-A1 Stabilized drug compositions WARNER-LAMBERT COMPANY (US) 1988-04-27 EP claimed
EP-0220107-A2 Use of angiotensin-converting enzyme inhibitors in macular degeneration MERCK & CO. INC. (US) 1987-04-29 EP claimed
US-4656188-A Ace inhibitors in macular degeneration MERCK & CO., INC. (US) 1987-04-07 US claimed