SCHEMBL15818924

SCHEMBL15818924

CC(C)(C)OC(=O)NCCCc1nc2c(Cl)cccc2c(=O)n1-c1cc(F)cc(F)c1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 4/20 0.40
DRD2 P14416 1/20 0.40
NQO2 P16083 1/20 0.39
STK17B O94768 1/20 0.39
STK17A Q9UEE5 1/20 0.39
PDE7A Q13946 2/20 0.39
ISG15 P05161 1/20 0.38
USP5 P45974 1/20 0.38
USP16 Q9Y5T5 1/20 0.38
USP3 Q9Y6I4 1/20 0.38
TLR7 Q9NYK1 4/20 0.38
BRD4 O60885 1/20 0.38
LMNA P02545 1/20 0.37
GAA P10253 1/20 0.37
HPGD P15428 1/20 0.37
PIK3CD O00329 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15819077 0.95 NQO2 (0.43) HDAC6DRD2NQO2STK17BSTK17A
SCHEMBL15819512 0.91 NQO2 (0.41) HDAC6NQO2TLR7BRD4PIK3CD
SCHEMBL15819594 0.90 BRD4 (0.40) HDAC6NQO2PDE7ATLR7BRD4
SCHEMBL15818376 0.86 PDE10A (0.45) DRD2STK17BSTK17ABRD4LMNA
SCHEMBL15818996 0.86 STK17B (0.38) DRD2STK17BSTK17ABRD4GAA
SCHEMBL15818820 0.86 PDE10A (0.48) LMNA
SCHEMBL15819206 0.86 PLK1 (0.39) NQO2STK17BSTK17ATLR7BRD4
SCHEMBL15818524 0.85 NQO2 (0.43) HDAC6NQO2PDE7ABRD4PIK3CD
SCHEMBL15820457 0.85 NQO2 (0.38) NQO2STK17BSTK17ABRD4LMNA
SCHEMBL15819357 0.84 NQO2 (0.47) HDAC6NQO2TLR7BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2935246-A1 ISOQUINOLINONE OR QUINAZOLINONE PHOSPHATIDYLINOSITOL 3-KINASE INHIBITORS Gilead Calistoga LLC (US) 2015-10-28 EP disclosed
WO-2014100767-A1 ISOQUINOLINONE OR QUINAZOLINONE PHOSPHATIDYLINOSITOL 3-KINASE INHIBITORS GILEAD CALISTOGA LLC (US) 2014-06-26 WO disclosed