SCHEMBL15909453

SCHEMBL15909453

CC(CN1CCc2oc(-c3ccc(OCc4ccc(C(F)(F)F)cc4)cc3)nc2C1)C(=O)O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
S1PR5 Q9H228 14/20 1.00
S1PR1 P21453 7/20 1.00
S1PR3 Q99500 6/20 1.00
PPARD Q03181 4/20 0.46
PPARG P37231 3/20 0.46
PPARA Q07869 2/20 0.46
ADAMTS4 O75173 1/20 0.45
MMP13 P45452 1/20 0.45
HRH3 Q9Y5N1 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15909566 0.89 S1PR5 (1.00) S1PR5S1PR1S1PR3PPARDPPARG
SCHEMBL15164300 0.76 S1PR5 (0.79) S1PR5S1PR1S1PR3
SCHEMBL3669682 0.74 S1PR5 (0.72) S1PR5S1PR1S1PR3
SCHEMBL18550025 0.73 S1PR5 (0.58) S1PR5S1PR1S1PR3PPARGADAMTS4
SCHEMBL320491 0.73 S1PR5 (1.00) S1PR5S1PR1S1PR3PPARGPPARA
SCHEMBL15909524 0.72 S1PR5 (0.67) S1PR5S1PR1S1PR3ADAMTS4MMP13
SCHEMBL6234038 0.71 PPARD (0.76) S1PR5S1PR1S1PR3PPARDPPARG
SCHEMBL15166548 0.71 S1PR5 (0.64) S1PR5S1PR1S1PR3
SCHEMBL18549817 0.71 S1PR5 (0.67) S1PR5S1PR1S1PR3PPARDPPARA
SCHEMBL322153 0.71 S1PR5 (0.68) S1PR5S1PR1S1PR3HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE48301-E1 Fused heterocyclic derivatives as S1P modulators ABBVIE B.V. (NL) 2020-11-10 US claimed
US-8796262-B2 Fused heterocyclic derivatives as S1P modulators ABBVIE B.V. (NL) 2014-08-05 US claimed
US-RE48301-E1 Fused heterocyclic derivatives as S1P modulators ABBVIE B.V. (NL) 2020-11-10 US disclosed
US-8796262-B2 Fused heterocyclic derivatives as S1P modulators ABBVIE B.V. (NL) 2014-08-05 US disclosed
US-8796262-B2 Fused heterocyclic derivatives as S1P modulators ABBVIE B.V. (NL) 2014-08-05 US disclosed