SCHEMBL15929246

SCHEMBL15929246

CCN(CC)C(=O)C1CCCN(CC(=O)NC(COCc2ccccc2)C(=O)Nc2ccc(Oc3ccc(F)cc3)cc2)C1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.54
S1PR1 P21453 7/20 0.53
ALDH1A1 P00352 3/20 0.49
HSD17B10 Q99714 1/20 0.43
POLB P06746 1/20 0.43
HPGD P15428 1/20 0.43
CCKBR P32239 1/20 0.42
RAB9A P51151 1/20 0.42
MEN1 O00255 1/20 0.41
LMNA P02545 1/20 0.41
ALOX15 P16050 1/20 0.41
TSHR P16473 1/20 0.41
KMT2A Q03164 1/20 0.41
DRD3 P35462 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12044679 1.00 KDM4E (0.54) KDM4ES1PR1ALDH1A1HSD17B10POLB
SCHEMBL27840733 0.88 S1PR1 (0.56) S1PR1ALDH1A1HPGDCCKBRMEN1
SCHEMBL1371682 0.88 S1PR1 (0.56) S1PR1ALDH1A1HPGDCCKBRMEN1
SCHEMBL1375018 0.85 S1PR1 (0.54) S1PR1CCKBR
SCHEMBL27923638 0.85 S1PR1 (0.54) S1PR1CCKBR
SCHEMBL1372404 0.85 S1PR1 (0.64) KDM4ES1PR1ALDH1A1HPGDMEN1
SCHEMBL1372408 0.85 S1PR1 (0.64) KDM4ES1PR1ALDH1A1HPGDMEN1
SCHEMBL1373075 0.84 S1PR1 (0.58) S1PR1ALDH1A1CCKBRMEN1LMNA
SCHEMBL1372392 0.84 S1PR1 (0.63) KDM4ES1PR1ALDH1A1HPGDMEN1
SCHEMBL13392746 0.84 S1PR1 (0.63) KDM4ES1PR1ALDH1A1HPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8802692-B2 Synergistic effects between sphingosine-1-phosphate receptor antagonists and antimicrotubule agents EXELIXIS, INC. (US) 2014-08-12 US claimed