SCHEMBL15933688

SCHEMBL15933688

c1cncc(-c2nc3n(n2)CCNC3)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 1/20 0.55
CD274 Q9NZQ7 1/20 0.55
CYP1A2 P05177 3/20 0.46
CYP3A4 P08684 3/20 0.46
ALOX15 P16050 2/20 0.46
CYP2D6 P10635 2/20 0.46
CLK4 Q9HAZ1 2/20 0.46
GBA1 P04062 1/20 0.46
MKNK1 Q9BUB5 1/20 0.44
MKNK2 Q9HBH9 1/20 0.44
TLR8 Q9NR97 1/20 0.42
TLR7 Q9NYK1 1/20 0.42
OGA O60502 1/20 0.41
ALDH1A1 P00352 3/20 0.41
HSD17B10 Q99714 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
KDM4E B2RXH2 1/20 0.41
LMNA P02545 1/20 0.41
TP53 P04637 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15933521 0.84 PDCD1 (0.69) PDCD1CD274TLR8TLR7ALDH1A1
SCHEMBL15933641 0.82 PDCD1 (0.53) PDCD1CD274TLR8TLR7
SCHEMBL5112559 0.82 PDCD1 (0.53) PDCD1CD274TLR8TLR7
SCHEMBL15933692 0.77 PDCD1 (0.57) PDCD1CD274ALOX15TLR8TLR7
SCHEMBL15933476 0.77 PDCD1 (0.48) PDCD1CD274CLK4TLR8TLR7
SCHEMBL15933679 0.77 PDCD1 (0.45) PDCD1CD274TLR8TLR7CHRNB2
SCHEMBL15933637 0.77 PDCD1 (0.57) PDCD1CD274TLR8TLR7NISCH
SCHEMBL15933639 0.77 PDCD1 (0.57) PDCD1CD274CYP1A2CYP3A4CYP2D6
SCHEMBL15933520 0.77 PDCD1 (0.64) PDCD1CD274CYP1A2TLR8TLR7
SCHEMBL15933685 0.75 PDCD1 (0.52) PDCD1CD274CYP1A2CYP2D6TLR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014117318-A1 NOVEL TRIAZOLE ANTIFUNGAL COMPOUNDS, AND PHARMACEUTICAL COMPOSITION, PREPARATION METHOD, AND APPLICATION THEREOF 中国科学院上海药物研究所 (CN) 2014-08-07 WO disclosed