SCHEMBL15934205

SCHEMBL15934205

Cc1noc(C2(C)CCCN2)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KRAS P01116 1/20 0.39
CHRM2 P08172 1/20 0.38
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36
HSD11B1 P28845 1/20 0.36
PARP1 P09874 7/20 0.33
PARP2 Q9UGN5 4/20 0.32
TNKS O95271 1/20 0.32
PARP14 Q460N5 1/20 0.32
PARP10 Q53GL7 1/20 0.32
PARP12 Q9H0J9 1/20 0.32
TNKS2 Q9H2K2 1/20 0.32
PARP4 Q9UKK3 1/20 0.32
PARP3 Q9Y6F1 1/20 0.32
CDC7 O00311 1/20 0.30
CCNE1 P24864 1/20 0.30
CDK2 P24941 1/20 0.30
ROCK1 Q13464 1/20 0.30
DBF4 Q9UBU7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15931994 0.80 PARP1 (0.33) PARP1PARP2TNKSPARP14PARP10
SCHEMBL21163476 0.77 POLB (0.38)
SCHEMBL16464351 0.76 HTT (0.48)
SCHEMBL16464352 0.76 HTT (0.48)
SCHEMBL16464353 0.76 HTT (0.48)
SCHEMBL13844344 0.72 CHRM2 (0.44) KRASCHRM2SLC6A2SLC6A4SLC6A3
Hydrochloric Acid SCHEMBL20292111 0.71 SLC6A2 (0.42) KRASCHRM2SLC6A2SLC6A4SLC6A3
SCHEMBL661466 0.70 SLC6A2 (0.41) KRASCHRM2SLC6A2SLC6A4SLC6A3
SCHEMBL661939 0.70 SLC6A2 (0.41) KRASCHRM2SLC6A2SLC6A4SLC6A3
SCHEMBL660453 0.70 SLC6A2 (0.41) KRASCHRM2SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20140221332-A1 METABOTROPHIC GLUTAMATE RECEPTOR 5 MODULATORS AND METHODS OF USE THEREOF SUNOVION PHARMACEUTICALS INC. (US) 2014-08-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140221332-A1 METABOTROPHIC GLUTAMATE RECEPTOR 5 MODULATORS AND METHODS OF USE THEREOF GRM5, GRIK5, GRM2 KRAS 3213/4885CHRM2 591/4885SLC6A2 442/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.