SCHEMBL15935754

SCHEMBL15935754

O=C(O)Cc1ccc(Oc2nc(-c3ccc(S)s3)nc3c2CCC3)cc1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 9/20 0.43
PDE4D Q08499 5/20 0.37
SRD5A2 P31213 2/20 0.37
RXRA P19793 3/20 0.35
RXRB P28702 3/20 0.35
RXRG P48443 3/20 0.35
BCHE P06276 2/20 0.35
ACHE P22303 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
LMNA P02545 1/20 0.34
THRB P10828 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15935758 0.89 PDE4B (0.44) PDE4BPDE4DSRD5A2RXRARXRB
SCHEMBL17290172 0.88 PDE4B (0.47) PDE4BPDE4DSRD5A2RXRARXRB
SCHEMBL15935755 0.88 PDE4B (0.44) PDE4BPDE4DSRD5A2RXRARXRB
SCHEMBL17290175 0.87 PDE4B (0.48) PDE4BPDE4DSRD5A2BCHEACHE
SCHEMBL15935818 0.86 PDE4B (0.42) PDE4BPDE4DSRD5A2RXRARXRB
SCHEMBL17290108 0.85 PDE4B (0.47) PDE4BPDE4DSRD5A2RXRARXRB
SCHEMBL15935753 0.85 PDE4B (0.41) PDE4BPDE4DSRD5A2RXRARXRB
SCHEMBL15935762 0.84 PDE4B (0.41) PDE4BPDE4DSRD5A2RXRARXRB
SCHEMBL15935752 0.82 PDE4B (0.42) PDE4BPDE4DSRD5A2RXRARXRB
SCHEMBL15935751 0.82 PDE4B (0.43) PDE4BPDE4DSRD5A2RXRARXRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014117948-A1 NOVEL SUBSTITUTED CONDENSED PYRIMIDINE COMPOUNDS Grünenthal GmbH (DE) 2014-08-07 WO disclosed