SCHEMBL15935987

SCHEMBL15935987

COc1ccc(CN2CCSc3ccccc3C2)cc1

nearest known ligand 0.61

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 5/20 0.55
TNF P01375 1/20 0.49
NOD2 Q9HC29 1/20 0.49
NOD1 Q9Y239 1/20 0.49
ABCB1 P08183 1/20 0.49
ABCC1 P33527 1/20 0.49
ABCG2 Q9UNQ0 1/20 0.49
ALDH1A1 P00352 1/20 0.47
POLB P06746 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
RYR2 Q92736 2/20 0.46
REV1 Q9UBZ9 1/20 0.45
CHKA P35790 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6867282 0.85 RYR2 (0.60) SIGMAR1ALDH1A1RYR2
SCHEMBL6867057 0.84 RYR2 (0.51) SIGMAR1RYR2
SCHEMBL15935957 0.83 DRD4 (0.51) SIGMAR1TNFNOD2NOD1ALDH1A1
SCHEMBL6868322 0.81 RYR2 (0.60) RYR2
SCHEMBL6867909 0.80 RYR2 (0.57) RYR2
SCHEMBL13302252 0.79 TNF (0.70) SIGMAR1TNFNOD2NOD1ABCB1
SCHEMBL15342814 0.77 RYR2 (0.54) RYR2
SCHEMBL15327766 0.77 RYR2 (0.54) RYR2
Surlorian SCHEMBL29728244 0.77 RYR2 (0.58) RYR2
Surlorian SCHEMBL15326996 0.77 RYR2 (0.58) RYR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2764867-A1 Agents for preventing and treating disorders Involving modulation of the RYR receptors The Trustees of Columbia University in the City of New York (US) 2014-08-13 EP claimed