SCHEMBL15949005

SCHEMBL15949005

Cc1ccccc1C(CC(=O)c1ccncc1)c1ccc(-c2cncnc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 3/20 0.49
CTSA P10619 8/20 0.42
HDAC4 P56524 1/20 0.41
MGAM O43451 1/20 0.40
GAA P10253 1/20 0.40
SI P14410 1/20 0.40
MGAM2 Q2M2H8 1/20 0.40
PLOD2 O00469 1/20 0.40
PLOD3 O60568 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
HPGD P15428 1/20 0.40
CYP2C19 P33261 1/20 0.40
PLOD1 Q02809 1/20 0.40
HIF1A Q16665 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.37
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15949092 0.88 GPBAR1 (0.62) GPBAR1CTSAHDAC4
SCHEMBL15949094 0.88 GPBAR1 (0.62) GPBAR1CTSAHDAC4
SCHEMBL15949109 0.87 HPGD (0.46) GPBAR1HDAC4PLOD2PLOD3ALDH1A1
SCHEMBL15949134 0.86 GPBAR1 (0.45) GPBAR1CTSAHDAC4
SCHEMBL363379 0.85 GPBAR1 (0.61) GPBAR1CTSAHDAC4GAA
SCHEMBL363055 0.85 GPBAR1 (0.61) GPBAR1CTSAHDAC4GAA
SCHEMBL362335 0.85 GPBAR1 (0.61) GPBAR1CTSAHDAC4GAA
SCHEMBL15949055 0.84 GPBAR1 (0.48) GPBAR1CTSAMGAMGAASI
SCHEMBL363384 0.83 MGAM (0.51) GPBAR1MGAMGAASIMGAM2
SCHEMBL361906 0.81 GPBAR1 (0.57) GPBAR1MGAMGAASIMGAM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-B1 1-HYDROXYIMINO-3-PHENYL-PROPANES HOFFMANN LA ROCHE (CH) 2014-08-20 EP claimed