SCHEMBL15949034

SCHEMBL15949034

COCCN(C)c1ccc(C(CC(=O)c2ccncc2)c2ccccc2C)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 3/20 0.42
L3MBTL1 Q9Y468 3/20 0.38
POLB P06746 1/20 0.38
HTT P42858 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
MGAM O43451 2/20 0.37
GAA P10253 2/20 0.37
SI P14410 2/20 0.37
MGAM2 Q2M2H8 2/20 0.37
CFTR P13569 1/20 0.36
CTSA P10619 2/20 0.36
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
TP53 P04637 1/20 0.36
USP1 O94782 1/20 0.36
DGAT1 O75907 1/20 0.35
PLOD2 O00469 1/20 0.35
PLOD3 O60568 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP1A2 P05177 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15948981 0.89 GPBAR1 (0.51) GPBAR1L3MBTL1MGAMGAASI
SCHEMBL15948980 0.89 GPBAR1 (0.51) GPBAR1L3MBTL1MGAMGAASI
SCHEMBL1389539 0.87 GPBAR1 (0.59) GPBAR1L3MBTL1NPSR1CFTRCTSA
SCHEMBL1389537 0.87 GPBAR1 (0.59) GPBAR1L3MBTL1NPSR1CFTRCTSA
SCHEMBL362837 0.87 GPBAR1 (0.59) GPBAR1L3MBTL1NPSR1CFTRCTSA
SCHEMBL361906 0.85 GPBAR1 (0.57) GPBAR1L3MBTL1POLBHTTNPSR1
SCHEMBL15949181 0.81 CNR2 (0.47) GPBAR1L3MBTL1POLBHTTNPSR1
SCHEMBL363384 0.78 MGAM (0.51) GPBAR1L3MBTL1POLBHTTNPSR1
SCHEMBL1389969 0.78 GPBAR1 (0.63) GPBAR1L3MBTL1NPSR1CFTRCTSA
SCHEMBL1389970 0.78 GPBAR1 (0.63) GPBAR1L3MBTL1NPSR1CFTRCTSA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-B1 1-HYDROXYIMINO-3-PHENYL-PROPANES HOFFMANN LA ROCHE (CH) 2014-08-20 EP claimed