SCHEMBL15949075

SCHEMBL15949075

Cc1cc(Cl)ccc1C(CC(=NO)c1ccc(=O)n(C)c1)c1ccc(-c2ccc(S(=O)(=O)O)cc2)cc1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 5/20 0.40
EGFR P00533 1/20 0.31
PPARG P37231 1/20 0.31
BRD4 O60885 1/20 0.31
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
ALOX15 P16050 1/20 0.30
CYP2C19 P33261 1/20 0.30
DRD2 P14416 1/20 0.30
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30
DRD3 P35462 1/20 0.30
HTR6 P50406 1/20 0.30
KEAP1 Q14145 1/20 0.30
NFE2L2 Q16236 1/20 0.30
FLT1 P17948 1/20 0.30
FLT4 P35916 1/20 0.30
KDR P35968 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15949073 1.00 GPBAR1 (0.40) GPBAR1EGFRPPARGBRD4CYP1A2
SCHEMBL1390699 0.92 GPBAR1 (0.40) GPBAR1CYP2D6
SCHEMBL10241381 0.92 GPBAR1 (0.40) GPBAR1CYP2D6
SCHEMBL10241383 0.92 GPBAR1 (0.40) GPBAR1CYP2D6
SCHEMBL370177 0.92 GPBAR1 (0.40) GPBAR1CYP2D6
SCHEMBL1389671 0.90 GPBAR1 (0.41) GPBAR1EGFRBRD4KEAP1NFE2L2
SCHEMBL368808 0.90 GPBAR1 (0.41) GPBAR1EGFRBRD4KEAP1NFE2L2
SCHEMBL1389674 0.90 GPBAR1 (0.41) GPBAR1EGFRBRD4KEAP1NFE2L2
SCHEMBL369333 0.90 GPBAR1 (0.41) GPBAR1EGFRBRD4KEAP1NFE2L2
SCHEMBL368806 0.90 GPBAR1 (0.41) GPBAR1EGFRBRD4KEAP1NFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-B1 1-HYDROXYIMINO-3-PHENYL-PROPANES HOFFMANN LA ROCHE (CH) 2014-08-20 EP disclosed