SCHEMBL15949124

SCHEMBL15949124

CCn1cc(C(=O)CC(c2ccc(Br)cc2)c2ccccc2C)ccc1=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 4/20 0.50
GAA P10253 4/20 0.43
MGAM O43451 3/20 0.43
SI P14410 3/20 0.43
MGAM2 Q2M2H8 3/20 0.43
KMT2A Q03164 3/20 0.38
APAF1 O14727 1/20 0.37
HSD17B10 Q99714 1/20 0.37
MAPT P10636 2/20 0.36
EPHX2 P34913 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
BRD4 O60885 1/20 0.35
BRD2 P25440 1/20 0.35
BRD3 Q15059 1/20 0.35
BRDT Q58F21 1/20 0.35
MEN1 O00255 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1390407 0.89 GPBAR1 (0.50) GPBAR1GAAMGAMSIMGAM2
SCHEMBL368424 0.89 GPBAR1 (0.48) GPBAR1GAAMGAMSIMGAM2
SCHEMBL369990 0.87 GPBAR1 (0.48) GPBAR1GAAMGAMSIMGAM2
SCHEMBL371067 0.87 GPBAR1 (0.46) GPBAR1GAAMGAMSIMGAM2
SCHEMBL1390266 0.87 GPBAR1 (0.48) GPBAR1GAAMGAMSIMGAM2
SCHEMBL369140 0.87 GPBAR1 (0.54) GPBAR1GAAMGAMSIMGAM2
SCHEMBL369733 0.87 GPBAR1 (0.54) GPBAR1GAAMGAMSIMGAM2
SCHEMBL369139 0.87 GPBAR1 (0.54) GPBAR1GAAMGAMSIMGAM2
SCHEMBL369091 0.87 GPBAR1 (0.62) GPBAR1GAAMGAMSIMGAM2
SCHEMBL370700 0.87 GPBAR1 (0.62) GPBAR1GAAMGAMSIMGAM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-B1 1-HYDROXYIMINO-3-PHENYL-PROPANES HOFFMANN LA ROCHE (CH) 2014-08-20 EP disclosed