SCHEMBL15958601

SCHEMBL15958601

COc1nc2ccsc2nc1-c1cccs1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 6/20 0.54
ADORA1 P30542 5/20 0.54
RPS6KB2 Q9UBS0 4/20 0.51
ALDH1A1 P00352 3/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
USP2 O75604 1/20 0.39
CYP1A2 P05177 1/20 0.39
GLA P06280 1/20 0.39
CYP3A4 P08684 1/20 0.39
GAA P10253 1/20 0.39
CYP2C9 P11712 1/20 0.39
CASP1 P29466 1/20 0.39
CASP7 P55210 1/20 0.39
HIF1A Q16665 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CLK4 Q9HAZ1 1/20 0.39
PDGFRB P09619 1/20 0.39
PDGFRA P16234 1/20 0.39
NPC1 O15118 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8225196 0.94 RPS6KB2 (0.55) ADORA2AADORA1RPS6KB2ALDH1A1MEN1
SCHEMBL7917553 0.84 ADORA2A (0.44) ADORA2AADORA1RPS6KB2ALDH1A1MEN1
SCHEMBL8380340 0.84 ADORA2A (0.50) ADORA2AADORA1RPS6KB2ALDH1A1MEN1
SCHEMBL8030948 0.83 RPS6KB2 (0.59) ADORA2AADORA1RPS6KB2ALDH1A1MEN1
SCHEMBL14164355 0.82 RPS6KB2 (0.59) ADORA2AADORA1RPS6KB2ALDH1A1MEN1
SCHEMBL8219378 0.80 RPS6KB2 (0.56) ADORA2AADORA1RPS6KB2ALDH1A1MEN1
SCHEMBL8211524 0.79 RPS6KB2 (0.82) ADORA2AADORA1RPS6KB2ALDH1A1MEN1
SCHEMBL7918132 0.78 RPS6KB2 (0.44) ADORA2AADORA1RPS6KB2ALDH1A1MEN1
SCHEMBL8381542 0.78 ADORA2A (0.50) ADORA2AADORA1RPS6KB2ALDH1A1MEN1
SCHEMBL24175690 0.78 HRH4 (0.38) ADORA2AADORA1RPS6KB2ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8809264-B2 Quinoxalinyl macrocyclic hepatitis C virus serine protease inhibitors ENANTA PHARMACEUTICALS, INC. (US) 2014-08-19 US disclosed