SCHEMBL15959004

SCHEMBL15959004

Bc1ccc([C@@H](C/C(Cc2ccncc2)=N\O)c2ccccc2C)cc1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 6/20 0.40
NR3C2 P08235 1/20 0.38
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34
GAA P10253 3/20 0.33
MAPT P10636 1/20 0.33
CHRM1 P11229 1/20 0.32
CYP19A1 P11511 1/20 0.32
CTSA P10619 1/20 0.32
ADRA2C P18825 1/20 0.32
LMNA P02545 1/20 0.31
TAAR1 Q96RJ0 1/20 0.31
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL362259 0.89 GPBAR1 (0.50) GPBAR1NR3C2GAAMAPTCYP19A1
SCHEMBL362261 0.89 GPBAR1 (0.50) GPBAR1NR3C2GAAMAPTCYP19A1
SCHEMBL363993 0.89 GPBAR1 (0.50) GPBAR1NR3C2GAAMAPTCYP19A1
SCHEMBL362260 0.89 GPBAR1 (0.50) GPBAR1NR3C2GAAMAPTCYP19A1
SCHEMBL1389694 0.84 GPBAR1 (0.60) GPBAR1NR3C2GAAMAPTCTSA
SCHEMBL1389695 0.84 GPBAR1 (0.60) GPBAR1NR3C2GAAMAPTCTSA
SCHEMBL364346 0.84 GPBAR1 (0.60) GPBAR1NR3C2GAAMAPTCTSA
SCHEMBL363855 0.84 GPBAR1 (0.60) GPBAR1NR3C2GAAMAPTCTSA
SCHEMBL1389692 0.84 GPBAR1 (0.60) GPBAR1NR3C2GAAMAPTCTSA
SCHEMBL15949123 0.81 GPBAR1 (0.46) GPBAR1NR3C2MAPTCYP19A1CTSA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-B1 1-HYDROXYIMINO-3-PHENYL-PROPANES HOFFMANN LA ROCHE (CH) 2014-08-20 EP disclosed