SCHEMBL15959593

SCHEMBL15959593

O=C(NC1=N[C@@]2(c3ccc(F)cc3F)COCC[C@H]2CS1)c1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.61
CYP2D6 P10635 2/20 0.42
KCNH2 Q12809 2/20 0.42
BACE2 Q9Y5Z0 3/20 0.42
CTSD P07339 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19218181 1.00 BACE1 (0.61) BACE1CYP2D6KCNH2BACE2CTSD
SCHEMBL12557551 0.91 BACE1 (0.61) BACE1CYP2D6KCNH2
SCHEMBL3302977 0.86 BACE1 (0.48) BACE1CYP2D6KCNH2BACE2CTSD
SCHEMBL3302981 0.86 BACE1 (0.48) BACE1CYP2D6KCNH2BACE2CTSD
SCHEMBL15839962 0.85 BACE1 (0.64) BACE1CYP2D6KCNH2BACE2CTSD
SCHEMBL15370009 0.85 BACE1 (0.43) BACE1CYP2D6KCNH2BACE2CTSD
SCHEMBL15839805 0.84 BACE1 (0.63) BACE1CYP2D6KCNH2BACE2CTSD
SCHEMBL15369977 0.84 BACE1 (0.50) BACE1CYP2D6KCNH2BACE2CTSD
SCHEMBL15940412 0.84 BACE1 (0.50) BACE1CYP2D6KCNH2BACE2CTSD
SCHEMBL15630253 0.84 BACE1 (0.63) BACE1KCNH2BACE2CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2956459-B1 SUBSTITUTED PHENYL-HEXAHYDROPYRANO[3,4-D][1,3]THIAZIN-2-AMINE COMPOUNDS PFIZER (US) 2017-07-19 EP disclosed
WO-2014125397-A1 SUBSTITUTED PHENYL HEXAHYDROPYRANO[3,4-d][1,3]THIAZIN-2-AMINE COMPOUNDS PFIZER INC. (US) 2014-08-21 WO disclosed