SCHEMBL15975809

SCHEMBL15975809

COc1ccc(-c2nn3c(-c4ccc(C#N)cc4)cnc3s2)cc1OC

nearest known ligand 0.77

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 5/20 0.77
FYN P06241 5/20 0.54
MKNK1 Q9BUB5 7/20 0.54
MKNK2 Q9HBH9 7/20 0.54
KDM4E B2RXH2 3/20 0.51
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
DCTPP1 Q9H773 1/20 0.51
ALDH1A1 P00352 2/20 0.50
USP2 O75604 1/20 0.50
LMNA P02545 1/20 0.50
TSHR P16473 1/20 0.50
MAPK1 P28482 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
HSD17B10 Q99714 1/20 0.50
PKM P14618 1/20 0.50
HPGD P15428 1/20 0.50
STAT6 P42226 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL532633 0.91 PIK3CA (0.74) PIK3CAFYNKDM4EMEN1KMT2A
SCHEMBL532016 0.87 PIK3CA (1.00) PIK3CAFYNKDM4EMEN1KMT2A
SCHEMBL2123322 0.83 PIK3CA (1.00) PIK3CAFYNKDM4EMEN1KMT2A
SCHEMBL15975812 0.82 PIK3CA (0.64) PIK3CAFYNKDM4EMEN1KMT2A
SCHEMBL15975807 0.80 PIK3CA (0.70) PIK3CAKDM4EMEN1KMT2ADCTPP1
SCHEMBL532334 0.80 PIK3CA (0.64) PIK3CAFYNKDM4EALDH1A1USP2
SCHEMBL532289 0.80 PIK3CA (0.67) PIK3CAFYNKDM4EMEN1KMT2A
SCHEMBL532748 0.79 PIK3CA (0.63) PIK3CAFYNKDM4EMEN1KMT2A
SCHEMBL25437299 0.79 MKNK1 (0.68) PIK3CAMKNK1MKNK2KDM4EMEN1
SCHEMBL532198 0.78 PIK3CA (0.61) PIK3CAFYNKDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8815918-B2 Imidazo [2, 1-B] [1, 3, 4] thiadiazole derivatives CENTRO NACIONAL DE INVESTIGACIONES ONCOLOGICAS (CNIO) (ES) 2014-08-26 US disclosed