SCHEMBL15975822

SCHEMBL15975822

COc1ccc(-c2nn3c(-c4cnc(C)nc4)c(C)nc3s2)cc1OC

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 6/20 0.80
ALDH1A1 P00352 6/20 0.53
KDM4E B2RXH2 5/20 0.53
MAPK1 P28482 5/20 0.53
TSHR P16473 3/20 0.53
HSD17B10 Q99714 3/20 0.53
LMNA P02545 2/20 0.53
NPSR1 Q6W5P4 2/20 0.53
USP2 O75604 1/20 0.53
DCTPP1 Q9H773 3/20 0.51
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
HPGD P15428 6/20 0.48
SIRT1 Q96EB6 1/20 0.48
KDM4C Q9H3R0 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
PKM P14618 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL532475 0.91 PIK3CA (0.77) PIK3CAALDH1A1KDM4EMAPK1TSHR
SCHEMBL532676 0.91 PIK3CA (0.79) PIK3CAALDH1A1KDM4EMAPK1TSHR
SCHEMBL532925 0.89 PIK3CA (1.00) PIK3CAALDH1A1KDM4EMAPK1TSHR
SCHEMBL533090 0.88 PIK3CA (0.79) PIK3CAALDH1A1KDM4EMAPK1TSHR
SCHEMBL533117 0.86 PIK3CA (0.76) PIK3CAALDH1A1KDM4EMAPK1TSHR
SCHEMBL15975819 0.86 PIK3CA (0.72) PIK3CAALDH1A1KDM4EMAPK1TSHR
SCHEMBL15975811 0.85 PIK3CA (0.71) PIK3CAALDH1A1KDM4EMAPK1TSHR
SCHEMBL532153 0.84 PIK3CA (0.72) PIK3CAALDH1A1KDM4EMAPK1TSHR
SCHEMBL15975807 0.82 PIK3CA (0.70) PIK3CAALDH1A1KDM4EMAPK1TSHR
SCHEMBL532283 0.82 PIK3CA (0.67) PIK3CAALDH1A1KDM4EMAPK1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8815918-B2 Imidazo [2, 1-B] [1, 3, 4] thiadiazole derivatives CENTRO NACIONAL DE INVESTIGACIONES ONCOLOGICAS (CNIO) (ES) 2014-08-26 US disclosed