SCHEMBL15975841

SCHEMBL15975841

CC(F)(F)c1cc(-c2cnc3sc(-c4cccc(S(C)(=O)=O)c4)nn23)cnc1N

nearest known ligand 0.88

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 11/20 0.88
KCNH2 Q12809 4/20 0.43
LOXL2 Q9Y4K0 1/20 0.40
NR1H2 P55055 2/20 0.39
NR1H3 Q13133 2/20 0.39
RXRA P19793 1/20 0.39
PRKDC P78527 1/20 0.38
ATM Q13315 1/20 0.38
ATR Q13535 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL533128 0.94 PIK3CA (1.00) PIK3CAKCNH2LOXL2NR1H2NR1H3
SCHEMBL15975826 0.86 PIK3CA (0.88) PIK3CAATR
SCHEMBL15975839 0.84 PIK3CA (0.66) PIK3CA
SCHEMBL15975816 0.84 PIK3CA (0.63) PIK3CA
SCHEMBL15975813 0.83 PIK3CA (0.71) PIK3CA
SCHEMBL15975829 0.83 PIK3CA (0.61) PIK3CA
SCHEMBL15975834 0.82 PIK3CA (0.67) PIK3CA
SCHEMBL2121274 0.81 PIK3CA (0.78) PIK3CAKCNH2
SCHEMBL452468 0.80 PIK3CA (1.00) PIK3CA
SCHEMBL15975842 0.79 PIK3CA (0.86) PIK3CAKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8815918-B2 Imidazo [2, 1-B] [1, 3, 4] thiadiazole derivatives CENTRO NACIONAL DE INVESTIGACIONES ONCOLOGICAS (CNIO) (ES) 2014-08-26 US disclosed