SCHEMBL16004303

SCHEMBL16004303

COc1ccc(C(=O)N2CCOc3ccc(COCCO)cc3C2)cc1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HPGD P15428 5/20 0.49
SMN1; SMN2 Q16637 3/20 0.49
PIK3CA P42336 7/20 0.44
GPR183 P32249 1/20 0.44
DRD2 P14416 2/20 0.43
DRD3 P35462 1/20 0.43
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
MAPT P10636 2/20 0.42
GAA P10253 1/20 0.42
RYR2 Q92736 1/20 0.42
LMNA P02545 1/20 0.41
KMT2A Q03164 1/20 0.41
RIPK1 Q13546 1/20 0.41
POLB P06746 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16004254 0.89 PIK3CA (0.47) HPGDSMN1; SMN2PIK3CAGPR183DRD2
SCHEMBL16004308 0.89 ABCB1 (0.48) HPGDSMN1; SMN2NPC1MAPTGAA
SCHEMBL16003999 0.88 PIK3CA (0.51) HPGDSMN1; SMN2PIK3CANPC1LMNA
SCHEMBL16004247 0.88 HPGD (0.51) HPGDSMN1; SMN2PIK3CAGPR183DRD2
SCHEMBL16004059 0.82 HPGD (0.47) HPGDSMN1; SMN2PIK3CAGPR183DRD2
SCHEMBL16004307 0.80 PIK3CA (0.40) PIK3CANPC1RAB9ARIPK1
SCHEMBL16003985 0.79 ATM (0.43) HPGDPIK3CAGAAKMT2ARIPK1
SCHEMBL17960292 0.79 HDAC6 (0.58) HPGDSMN1; SMN2PIK3CAGPR183NPC1
SCHEMBL16003975 0.79 ABCB1 (0.46) HPGDSMN1; SMN2NPC1RAB9AMAPT
SCHEMBL16004248 0.78 ABCB1 (0.50) HPGDSMN1; SMN2NPC1MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014133414-A2 HETEROCYCLIC TGR5 BILE ACID RECEPTOR AGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR THE PRODUCTION AND USE THEREOF АЛЛА ХЕМ ЛЛС (US) 2014-09-04 WO disclosed