SCHEMBL16008362

SCHEMBL16008362

CCOC(=O)c1cc2c(-c3cc(NS(C)(=O)=O)ccc3Oc3ccc(F)cc3F)[nH]c(C)c2c(=O)[nH]1

nearest known ligand 0.66

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 19/20 0.66
EP300 Q09472 1/20 0.48
MMP2 P08253 1/20 0.46
MMP13 P45452 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16007975 0.94 BRD4 (0.59) BRD4EP300
SCHEMBL16007942 0.89 BRD4 (0.69) BRD4EP300
SCHEMBL16007895 0.88 BRD4 (0.65) BRD4
SCHEMBL16008027 0.88 BRD4 (0.49) BRD4
SCHEMBL16008085 0.86 BRD4 (0.49) BRD4
SCHEMBL16007275 0.86 BRD4 (0.51) BRD4EP300
SCHEMBL16007965 0.86 BRD4 (0.66) BRD4MMP2MMP13
SCHEMBL16007910 0.86 BRD4 (0.51) BRD4
SCHEMBL16008135 0.83 BRD4 (0.48) BRD4
SCHEMBL16149004 0.81 BRD4 (0.54) BRD4EP300

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9050346-B2 Bromodomain inhibitors ABBVIE INC. (US) 2015-06-09 US claimed
US-20140256705-A1 BROMODOMAIN INHIBITORS ABBVIE INC. 2014-09-11 US claimed
US-9050346-B2 Bromodomain inhibitors ABBVIE INC. (US) 2015-06-09 US disclosed
US-20140256705-A1 BROMODOMAIN INHIBITORS ABBVIE INC. 2014-09-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140256705-A1 BROMODOMAIN INHIBITORS BRD4, BRD3, BRD1 BRD4 1/4885EP300 14/4885MMP2 1297/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.