SCHEMBL16016121

SCHEMBL16016121

Nc1cccc(C(=O)N=O)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PBRM1 Q86U86 1/20 0.57
NPC1 O15118 2/20 0.49
MITF O75030 1/20 0.49
LMNA P02545 1/20 0.49
POLB P06746 1/20 0.49
F2 P00734 1/20 0.48
PLG P00747 1/20 0.48
PRSS1 P07477 1/20 0.48
PRSS2 P07478 1/20 0.48
PRSS3 P35030 1/20 0.48
HDAC3 O15379 1/20 0.46
HDAC4 P56524 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC7 Q8WUI4 1/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC10 Q969S8 1/20 0.46
HDAC11 Q96DB2 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
HDAC9 Q9UKV0 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28924563 0.79 PBRM1 (0.52) PBRM1NPC1MITFLMNAPOLB
SCHEMBL125621 0.78 PBRM1 (0.87) PBRM1NPC1MITFLMNAPOLB
SCHEMBL9282073 0.78 PBRM1 (0.87) PBRM1NPC1MITFLMNAPOLB
SCHEMBL5091376 0.78 PBRM1 (0.65) PBRM1NPC1MITFLMNAPOLB
SCHEMBL29363032 0.78 PBRM1 (0.87) PBRM1NPC1MITFLMNAPOLB
SCHEMBL3981731 0.77 PBRM1 (0.50) PBRM1NPC1MITFLMNAPOLB
SCHEMBL8776892 0.77 PBRM1 (0.50) PBRM1NPC1MITFLMNAPOLB
SCHEMBL8003710 0.77 PBRM1 (0.59) PBRM1NPC1MITFLMNAPOLB
3-Aminobenzoic Acid SCHEMBL27648 0.76 PBRM1 (0.69) PBRM1NPC1MITFLMNAPOLB
3-Aminobenzamide SCHEMBL16070 0.76 PBRM1 (0.63) PBRM1NPC1MITFLMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2563123-B1 NOVEL BETA 3 ADRENERGIC RECEPTOR AGONISTS MERCK SHARP & DOHME (US) 2018-04-25 EP disclosed
WO-2018053353-A1 KETONE INHIBITORS OF LYSINE GINGIPAIN Cortexyme, Inc. (US) 2018-03-22 WO disclosed
EP-1809601-B1 COMPOUNDS FOR ALZHEIMER'S DISEASE MANFREDI JOHN (US) 2014-09-10 EP disclosed