SCHEMBL16052004

SCHEMBL16052004

CC1(c2ccc(OC(F)(F)F)cc2)CSC(N)=N1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 8/20 0.51
SLC6A4 P31645 8/20 0.43
SLC6A3 Q01959 6/20 0.42
SLC6A2 P23975 1/20 0.42
CTSD P07339 2/20 0.41
BACE2 Q9Y5Z0 2/20 0.41
KCNH2 Q12809 1/20 0.36
KDM1A O60341 1/20 0.35
RCOR1 Q9UKL0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10156776 0.86 BACE1 (0.71) BACE1SLC6A4SLC6A3SLC6A2BACE2
SCHEMBL5330236 0.75 BACE1 (0.70) BACE1KCNH2
SCHEMBL3617743 0.74 TAAR1 (0.60) BACE1
SCHEMBL3617749 0.74 TAAR1 (0.60) BACE1
SCHEMBL10154760 0.71 BACE1 (0.49) BACE1SLC6A4SLC6A3SLC6A2KCNH2
SCHEMBL28172966 0.69 SLC6A4 (0.49) BACE1SLC6A4SLC6A3SLC6A2CTSD
SCHEMBL5052720 0.69 BACE1 (0.65) BACE1KCNH2KDM1A
SCHEMBL12350637 0.68 BACE1 (0.76) BACE1CTSDBACE2KCNH2
SCHEMBL10195094 0.68 BACE1 (1.00) BACE1KCNH2
SCHEMBL10194679 0.68 SLC6A4 (0.54) SLC6A4SLC6A3SLC6A2KCNH2KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970255-A1 COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF INFLAMMATORY DISORDERS Galapagos NV (BE) 2016-01-20 EP claimed
WO-2014139882-A1 COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF INFLAMMATORY DISORDERS GALAPAGOS NV (BE) 2014-09-18 WO claimed