SCHEMBL16064992

SCHEMBL16064992

CNC(=O)NCCc1nccn1Cc1ccccc1Cl

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 11/20 0.56
HSP90B1 P14625 11/20 0.56
TP53 P04637 2/20 0.45
CNR1 P21554 1/20 0.44
BRD4 O60885 1/20 0.44
MTNR1A P48039 1/20 0.43
ADRA2C P18825 1/20 0.42
PTGER3 P43115 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
HSP90AB1 P08238 1/20 0.41
LMNA P02545 1/20 0.41
MAP3K14 Q99558 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16136365 0.88 HSP90AA1 (0.58) HSP90AA1HSP90B1TP53BRD4ADRA2C
SCHEMBL16133643 0.85 HSP90AA1 (0.55) HSP90AA1HSP90B1TP53BRD4ADRA2C
SCHEMBL20625806 0.84 HSP90AA1 (0.53) HSP90AA1HSP90B1TP53BRD4ADRA2C
SCHEMBL16768685 0.81 HSP90AA1 (0.50) HSP90AA1HSP90B1TP53BRD4ADRA2C
SCHEMBL16136339 0.79 HSP90AA1 (0.54) HSP90AA1HSP90B1TP53BRD4ADRA2C
SCHEMBL16133634 0.76 HSP90AA1 (0.52) HSP90AA1HSP90B1TP53BRD4ADRA2C
SCHEMBL6959787 0.75 HSP90AA1 (0.53) HSP90AA1HSP90B1LMNA
SCHEMBL19413280 0.75 HSP90AA1 (0.47) HSP90AA1HSP90B1TP53BRD4HSP90AB1
SCHEMBL16136314 0.73 HSP90AA1 (0.54) HSP90AA1HSP90B1HSP90AB1LMNA
SCHEMBL12851364 0.71 NPC1 (0.79) NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014144747-A1 SUBSTITUTED 6,5-FUSED BICYCLIC HETEROARYL COMPOUNDS Epizyme, Inc. (US) 2014-09-18 WO disclosed