SCHEMBL16065409

SCHEMBL16065409

Cc1cc(Nc2cc(N3CCOCC3)nc(Oc3ccc4[nH]c(C)cc4c3Cl)n2)n[nH]1

nearest known ligand 0.57

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PIK3C3 Q8NEB9 2/20 0.57
AURKA O14965 6/20 0.51
AURKB Q96GD4 2/20 0.51
EGFR P00533 8/20 0.49
TBK1 Q9UHD2 1/20 0.46
IGF1R P08069 2/20 0.46
RIPK1 Q13546 1/20 0.45
JAK3 P52333 1/20 0.44
NTRK1 P04629 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16065657 0.91 EGFR (0.61) PIK3C3AURKAAURKBEGFRTBK1
SCHEMBL15705010 0.91 EGFR (0.50) PIK3C3AURKAAURKBEGFRTBK1
SCHEMBL15705036 0.90 PIK3C3 (0.48) PIK3C3AURKAAURKBEGFRTBK1
SCHEMBL15704753 0.90 IGF1R (0.49) PIK3C3AURKAAURKBEGFRIGF1R
SCHEMBL17175935 0.90 EGFR (0.53) PIK3C3AURKAAURKBEGFRTBK1
SCHEMBL17175910 0.90 PIK3C3 (0.57) PIK3C3AURKAAURKBEGFRTBK1
SCHEMBL15705081 0.89 EGFR (0.49) PIK3C3AURKAAURKBEGFRTBK1
SCHEMBL17176002 0.89 EGFR (0.51) PIK3C3AURKAAURKBEGFRTBK1
SCHEMBL15705025 0.88 EGFR (0.51) PIK3C3AURKAAURKBEGFRTBK1
SCHEMBL16065567 0.88 EGFR (0.51) PIK3C3AURKAAURKBEGFRTBK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10245261-B2 Substituted indol-5-ol derivatives and their therapeutic applications NANTBIO, INC. (US) 2019-04-02 US disclosed
US-20170189400-A1 SUBSTITUTED INDOL-5-OL DERIVATIVES AND THEIR THERAPEUTIC APPLICATIONS NANTBIO, INC. 2017-07-06 US disclosed
US-20170088544-A1 SUBSTITUTED INDOL-5-OL DERIVATIVES AND THEIR THERAPEUTICAL APPLICATIONS NANTBIO, INC. 2017-03-30 US disclosed
US-9550760-B2 Substituted indol-5-ol derivatives and their therapeutic applications NANTBIOSCIENCE, INC. (US) 2017-01-24 US disclosed
US-9458137-B2 Substituted indol-5-ol derivatives and their therapeutical applications NANTBIOSCIENCE, INC. (US) 2016-10-04 US disclosed
US-20160016945-A1 SUBSTITUTED INDOL-5-OL DERIVATIVES AND THEIR THERAPEUTIC APPLICATIONS NANTBIO, INC. 2016-01-21 US disclosed
US-20150291564-A1 SUBSTITUTED INDOL-5-OL DERIVATIVES AND THEIR THERAPEUTICAL APPLICATIONS NANTBIOSCIENCE, INC. (US) 2015-10-15 US disclosed
WO-2014145403-A1 SUBSTITUTED INDOL-5-OL DERIVATIVES AND THEIR THERAPEUTIC APPLICATIONS NANTBIO, INC. (US) 2014-09-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170189400-A1 SUBSTITUTED INDOL-5-OL DERIVATIVES AND THEIR THERAPEUTIC APPLICATIONS GRK5, GRK3, CDK5 PIK3C3 507/4885AURKA 796/4885AURKB 406/4885
US-20170088544-A1 SUBSTITUTED INDOL-5-OL DERIVATIVES AND THEIR THERAPEUTICAL APPLICATIONS GRK5, GRK3, MTMR1 PIK3C3 471/4885AURKA 1063/4885AURKB 468/4885
US-10245261-B2 Substituted indol-5-ol derivatives and their therapeutic applications GRK5, GRK3, CDK5 PIK3C3 507/4885AURKA 796/4885AURKB 406/4885
US-20150291564-A1 SUBSTITUTED INDOL-5-OL DERIVATIVES AND THEIR THERAPEUTICAL APPLICATIONS GRK5, GRK3, MTMR1 PIK3C3 471/4885AURKA 1063/4885AURKB 468/4885
US-20160016945-A1 SUBSTITUTED INDOL-5-OL DERIVATIVES AND THEIR THERAPEUTIC APPLICATIONS GRK5, GRK3, CDK5 PIK3C3 507/4885AURKA 796/4885AURKB 406/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.