SCHEMBL16087219

SCHEMBL16087219

O=C(O)c1cc(-c2cnn3cc(-c4cccnc4)cnc23)cs1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MARK3 P27448 12/20 0.70
KDR P35968 8/20 0.54
FLT1 P17948 3/20 0.49
FLT4 P35916 3/20 0.49
ULK1 O75385 1/20 0.49
ULK2 Q8IYT8 1/20 0.49
MKNK2 Q9HBH9 1/20 0.49
STK17A Q9UEE5 1/20 0.49
SGK1 O00141 1/20 0.48
PIK3CD O00329 1/20 0.48
CHEK1 O14757 1/20 0.48
MAPK13 O15264 1/20 0.48
PDPK1 O15530 1/20 0.48
NUAK1 O60285 1/20 0.48
CCNT1 O60563 1/20 0.48
JAK2 O60674 1/20 0.48
ROCK2 O75116 1/20 0.48
CHEK2 O96017 1/20 0.48
EGFR P00533 1/20 0.48
RAF1 P04049 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3763532 0.99 MARK3 (0.69) MARK3KDRFLT1FLT4ULK1
SCHEMBL3772483 0.90 MARK3 (0.69) MARK3KDRFLT1FLT4ULK1
SCHEMBL5414309 0.88 KDR (0.60) MARK3KDRFLT1FLT4ULK1
SCHEMBL3762774 0.86 MARK3 (0.72) MARK3KDRULK1ULK2MKNK2
SCHEMBL3772433 0.85 MARK3 (0.70) MARK3KDRULK1ULK2MKNK2
SCHEMBL3766784 0.84 MARK3 (0.69) MARK3KDRULK1ULK2MKNK2
SCHEMBL3769325 0.83 MARK3 (0.70) MARK3KDRULK1ULK2MKNK2
SCHEMBL3766751 0.83 MARK3 (0.70) MARK3KDRULK1ULK2MKNK2
SCHEMBL3764916 0.83 MARK3 (0.68) MARK3KDRULK1ULK2MKNK2
SCHEMBL3769144 0.83 MARK3 (0.68) MARK3KDRULK1ULK2MKNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2178375-B1 PYRAZOLOÝ1,5-A¨PYRIMIDINE DERIVATIVES MERCK SHARP & DOHME (US) 2014-09-24 EP disclosed