SCHEMBL16144183

SCHEMBL16144183

CC(=O)c1cccc(C)c1-c1ccccn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.47
CTNNB1 P35222 1/20 0.45
WNT3A P56704 1/20 0.45
MYC P01106 1/20 0.45
GRM5 P41594 1/20 0.43
KDM4C Q9H3R0 1/20 0.43
MAPK1 P28482 2/20 0.43
BRD4 O60885 1/20 0.42
BRD2 P25440 1/20 0.42
BRD3 Q15059 1/20 0.42
BAZ2B Q9UIF8 1/20 0.42
BAZ2A Q9UIF9 1/20 0.42
KDM4E B2RXH2 3/20 0.42
LMNA P02545 2/20 0.42
CCR1 P32246 2/20 0.42
CCR5 P51681 2/20 0.42
CCR8 P51685 2/20 0.42
CYP1A2 P05177 1/20 0.42
POLB P06746 1/20 0.42
METAP1 P53582 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6876765 0.87 MYC (0.57) ALDH1A1CTNNB1WNT3AMYCKDM4C
SCHEMBL4726132 0.80 KDM4E (0.59) ALDH1A1GRM5MAPK1KDM4ELMNA
SCHEMBL30824691 0.80 KDM4E (0.59) ALDH1A1GRM5MAPK1KDM4ELMNA
SCHEMBL9200058 0.77 KDM4C (0.62) ALDH1A1GRM5KDM4CBRD4BRD2
SCHEMBL20903172 0.76 CBFB (0.38) CTNNB1WNT3AMYCGRM5MAPK1
SCHEMBL21562543 0.76 NPC1 (0.41) CTNNB1WNT3AMYCGRM5MAPK1
SCHEMBL18202141 0.76 PTPN1 (0.48) ALDH1A1MAPK1KDM4ELMNAPOLB
SCHEMBL14670506 0.76 KDM4E (0.48) ALDH1A1GRM5KDM4CBRD4BRD2
SCHEMBL2943452 0.75 GRM5 (0.54) ALDH1A1GRM5KDM4CMAPK1KDM4E
SCHEMBL21562542 0.75 GRM5 (0.39) CTNNB1WNT3AGRM5MAPK1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014159591-A1 SUBSTITUTED 7-AZABICYCLES AND THEIR USE AS OREXIN RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2014-10-02 WO disclosed