SCHEMBL16158593

SCHEMBL16158593

COC(=O)c1cc2c(cc1OC)CN(Cc1cccc(-n3ccc4ccccc43)c1)C(C)C2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMO Q99835 1/20 0.39
DRD2 P14416 5/20 0.38
DRD4 P21917 5/20 0.38
PTGER2 P43116 1/20 0.37
FGFR1 P11362 1/20 0.36
SRC P12931 1/20 0.36
MAPK14 Q16539 2/20 0.36
ALDH1A1 P00352 2/20 0.36
LMNA P02545 2/20 0.36
HPGD P15428 2/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
ABCB1 P08183 1/20 0.35
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34
USP2 O75604 1/20 0.34
MAPK1 P28482 1/20 0.34
PTK2 Q05397 3/20 0.34
KDM4E B2RXH2 1/20 0.34
ABCG2 Q9UNQ0 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16158588 0.90 ABCB1 (0.42) SMOPTGER2ABCB1CA2CA9
SCHEMBL17531438 0.85 FGFR1 (0.49) PTGER2FGFR1SRCRAB9A
SCHEMBL16147263 0.85 FGFR1 (0.49) PTGER2FGFR1SRCRAB9A
SCHEMBL17531469 0.78 FGFR1 (0.42) PTGER2FGFR1SRC
SCHEMBL16148304 0.78 FGFR1 (0.42) PTGER2FGFR1SRC
SCHEMBL16147266 0.75 KMT2A (0.45) MAPK14ALDH1A1LMNAHPGDNPC1
SCHEMBL16147349 0.74 FGFR1 (0.49) PTGER2FGFR1SRCCA2CA9
SCHEMBL17531428 0.74 FGFR1 (0.49) PTGER2FGFR1SRCCA2CA9
SCHEMBL17531440 0.72 FGFR1 (0.45) PTGER2FGFR1SRCCA2CA9
SCHEMBL16158445 0.72 HCRTR1 (0.38) PTGER2ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014165815-A2 NONSTEROIDAL AND STEROIDAL COMPOUNDS WITH POTENT ANDROGEN RECEPTOR DOWN-REGULATION AND ANTI PROSTATE CANCER ACTIVITY UNIVERSITY OF MARYLAND, BALTIMORE (US) 2014-10-09 WO disclosed