SCHEMBL16161908

SCHEMBL16161908

O=C(Nc1c(F)ccc(NS(=O)(=O)c2ccc(C(F)(F)F)cc2)c1F)Oc1cnc2[nH]cnc2c1

nearest known ligand 0.45

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BRAF P15056 3/20 0.45
CYP2C9 P11712 6/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C19 P33261 7/20 0.41
CYP3A4 P08684 7/20 0.40
CCR9 P51686 1/20 0.38
KDM1A O60341 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16162081 0.93 CCR9 (0.39) BRAFCYP2C9CCR9
SCHEMBL16162085 0.88 CYP2C19 (0.44) BRAFCYP2C9CYP2C19CYP3A4CCR9
SCHEMBL16162040 0.88 KIT (0.40) BRAFCYP2C9CYP2C19CCR9
SCHEMBL16162153 0.87 BRAF (0.44) BRAFCYP2C9CYP2D6CYP2C19CYP3A4
SCHEMBL16162111 0.86 CYP3A4 (0.46) BRAFCYP2C9CYP2C19CYP3A4
SCHEMBL16162106 0.86 CYP3A4 (0.47) BRAFCYP2C9CYP2C19CYP3A4
SCHEMBL300408 0.85 BRAF (0.46) BRAFCYP2C9CYP2D6CYP2C19CYP3A4
SCHEMBL16162083 0.85 BRAF (0.43) BRAFCYP2C9CYP3A4
SCHEMBL16162113 0.85 BRAF (0.48) BRAFCYP2C9CYP3A4
SCHEMBL16162151 0.84 CYP2D6 (0.43) BRAFCYP2C9CYP2D6CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2170830-B1 2-FLUORO-BENZENESULFONAMIDE COMPOUNDS AS Raf KINASE MODULATORS PLEXXIKON INC (US) 2014-10-15 EP claimed