SCHEMBL16162183

SCHEMBL16162183

CC(Nc1cnc2cc(-c3cnn(C(=O)OC(C)(C)C)c3)ccc2n1)c1cccc(N2CCN(C)CC2)c1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 3/20 0.41
DYRK1A Q13627 3/20 0.41
WNT1 P04628 2/20 0.41
ROCK2 O75116 1/20 0.38
MET P08581 2/20 0.38
TBK1 Q9UHD2 8/20 0.37
LRRK2 Q5S007 1/20 0.37
JAK3 P52333 1/20 0.36
PFKFB3 Q16875 3/20 0.36
ABL1 P00519 1/20 0.36
NTRK1 P04629 1/20 0.36
YES1 P07947 1/20 0.36
MAPK1 P28482 1/20 0.36
AURKB Q96GD4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL781221 1.00 GSK3B (0.41) GSK3BDYRK1AWNT1ROCK2MET
SCHEMBL781950 0.86 SCD (0.40) GSK3BDYRK1AROCK2TBK1PFKFB3
SCHEMBL780128 0.85 PFKFB3 (0.38) ROCK2TBK1PFKFB3MAPK1
SCHEMBL781210 0.85 FGFR4 (0.44) GSK3BROCK2PFKFB3
SCHEMBL780503 0.79 PFKFB3 (0.43) GSK3BDYRK1AWNT1ROCK2TBK1
SCHEMBL782116 0.79 AOC3 (0.41) GSK3BDYRK1AWNT1ROCK2MET
Hydrochloric Acid SCHEMBL16161587 0.78 PFKFB3 (0.42) GSK3BDYRK1AWNT1ROCK2TBK1
SCHEMBL27868791 0.76 KCNH2 (0.43) JAK3PFKFB3
SCHEMBL780785 0.76 KCNH2 (0.43) JAK3PFKFB3
SCHEMBL781898 0.72 MAPK1 (0.47) GSK3BDYRK1AWNT1ROCK2MET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2435423-B1 SUBSTITUTED BENZOTRIAZINES AND QUINOXALINES AS INHIBITORS OF P70S6 KINASE SENTINEL ONCOLOGY LTD (GB) 2014-10-15 EP disclosed