SCHEMBL16175409

SCHEMBL16175409

CS(=O)(=O)NC(=O)c1cc(Cl)c(Oc2cnc(C3CCC3)c(Cl)c2)cc1F

nearest known ligand 0.93

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 20/20 0.93
SCN2B O60939 1/20 0.93
SCN1A P35498 1/20 0.93
SCN1B Q07699 1/20 0.93
SCN5A Q14524 1/20 0.93

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1690140 0.96 SCN9A (1.00) SCN9ASCN2BSCN1ASCN1BSCN5A
SCHEMBL16175285 0.90 SCN9A (0.89) SCN9ASCN2BSCN1ASCN1BSCN5A
SCHEMBL16175332 0.89 SCN9A (0.83) SCN9ASCN2BSCN1ASCN1BSCN5A
SCHEMBL16174929 0.89 SCN9A (0.86) SCN9ASCN2BSCN1ASCN1BSCN5A
SCHEMBL1690203 0.87 SCN9A (0.83) SCN9ASCN2BSCN1ASCN1BSCN5A
SCHEMBL16175578 0.86 SCN9A (0.81) SCN9ASCN2BSCN1ASCN1BSCN5A
SCHEMBL370118 0.86 SCN9A (0.81) SCN9ASCN2BSCN1ASCN1BSCN5A
SCHEMBL16175181 0.85 SCN9A (0.80) SCN9ASCN2BSCN1ASCN1BSCN5A
SCHEMBL16175247 0.85 SCN9A (0.80) SCN9ASCN2BSCN1ASCN1BSCN5A
SCHEMBL369585 0.85 SCN9A (0.79) SCN9ASCN2BSCN1ASCN1BSCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593432-B1 N-SULFONYLBENZAMIDE DERIVATIVES USEFUL AS VOLTAGE GATED SODIUM CHANNEL INHIBITORS PFIZER LTD (GB) 2014-10-22 EP disclosed