SCHEMBL16181797

SCHEMBL16181797

CCCCCCNCC(F)(F)F

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.55
ALDH1A1 P00352 1/20 0.55
EPHX1 P07099 8/20 0.45
ADH1B P00325 1/20 0.44
ADH1C P00326 1/20 0.44
ADH1A P07327 1/20 0.44
ADH4 P08319 1/20 0.44
ADH7 P40394 1/20 0.44
S1PR2 O95136 5/20 0.41
S1PR4 O95977 5/20 0.41
S1PR1 P21453 5/20 0.41
S1PR3 Q99500 5/20 0.41
S1PR5 Q9H228 1/20 0.41
THRB P10828 1/20 0.38
HRH4 Q9H3N8 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
ANPEP P15144 1/20 0.36
ERAP2 Q6P179 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10688479 1.00 TSHR (0.55) TSHRALDH1A1EPHX1ADH1BADH1C
SCHEMBL10686025 1.00 TSHR (0.55) TSHRALDH1A1EPHX1ADH1BADH1C
SCHEMBL10687887 1.00 TSHR (0.55) TSHRALDH1A1EPHX1ADH1BADH1C
SCHEMBL10686612 1.00 TSHR (0.55) TSHRALDH1A1EPHX1ADH1BADH1C
SCHEMBL10687034 1.00 TSHR (0.55) TSHRALDH1A1EPHX1ADH1BADH1C
SCHEMBL11324424 0.98 TSHR (0.57) TSHRALDH1A1EPHX1ADH1BADH1C
SCHEMBL2608049 0.90 TSHR (0.50) TSHRALDH1A1EPHX1ADH1BADH1C
SCHEMBL15114026 0.84 TSHR (0.52) TSHRALDH1A1EPHX1ADH1BADH1C
SCHEMBL15114057 0.84 TSHR (0.52) TSHRALDH1A1EPHX1ADH1BADH1C
SCHEMBL15114072 0.84 TSHR (0.52) TSHRALDH1A1EPHX1ADH1BADH1C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2170848-B1 PYRAZINONE DERIVATIVES AND THEIR USE IN THE TREATMENT OF LUNG DISEASES ASTRAZENECA AB (SE) 2014-10-22 EP disclosed