SCHEMBL16189192

SCHEMBL16189192

Cc1cnc2c(c1)NNN2c1ccc(C(=O)N(c2ncccc2Cl)[C@@H]2CCCNC2)nc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PCSK9 Q8NBP7 16/20 0.69
RPLP1 P05386 12/20 0.69
RPLP0 P05388 12/20 0.69
RPS17 P08708 12/20 0.69
RPSA P08865 12/20 0.69
RPS2 P15880 12/20 0.69
RPL35A P18077 12/20 0.69
RPL7 P18124 12/20 0.69
RPL17 P18621 12/20 0.69
RPS4Y1 P22090 12/20 0.69
RPS3 P23396 12/20 0.69
RPS12 P25398 12/20 0.69
RPL13 P26373 12/20 0.69
RPL10 P27635 12/20 0.69
RPL12 P30050 12/20 0.69
RPL9; RPL9P7; RPL9P8; RPL9P9 P32969 12/20 0.69
RPL22 P35268 12/20 0.69
RPL4 P36578 12/20 0.69
RPS19 P39019 12/20 0.69
RPL3 P39023 12/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16189119 0.91 PCSK9 (0.68) PCSK9RPLP1RPLP0RPS17RPSA
SCHEMBL16177345 0.81 PCSK9 (1.00) PCSK9RPLP1RPLP0RPS17RPSA
SCHEMBL24176583 0.81 PCSK9 (0.64) PCSK9RPLP1RPLP0RPS17RPSA
SCHEMBL16177805 0.76 PCSK9 (1.00) PCSK9RPLP1RPLP0RPS17RPSA
SCHEMBL16177128 0.74 PCSK9 (1.00) PCSK9RPLP1RPLP0RPS17RPSA
SCHEMBL24756398 0.73 PCSK9 (0.64) PCSK9RPLP1RPLP0RPS17RPSA
SCHEMBL17669169 0.69 PCSK9 (0.86) PCSK9RPLP1RPLP0RPS17RPSA
SCHEMBL17679154 0.69 PCSK9 (0.66) PCSK9RPLP1RPLP0RPS17RPSA
SCHEMBL16177066 0.67 PCSK9 (0.74) PCSK9RPLP1RPLP0RPS17RPSA
SCHEMBL16180190 0.66 PCSK9 (0.81) PCSK9RPLP1RPLP0RPS17RPSA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014170786-A1 N-PIPERIDIN-3-YLBENZAMIDE DERIVATIVES FOR TREATING CARDIOVASCULAR DISEASES PFIZER INC. (US) 2014-10-23 WO disclosed