SCHEMBL16199019

SCHEMBL16199019

Cc1cc(C(=O)N[C@@H]2CCCC(Nc3nc(-c4n[nH]c5ncc(F)cc45)ncc3F)C2)cs1

nearest known ligand 0.54

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 2/20 0.38
GSK3B P49841 2/20 0.38
FLT3 P36888 2/20 0.38
JAK2 O60674 1/20 0.38
SRC P12931 1/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16199078 0.91 GSK3A (0.38) GSK3AGSK3BFLT3
SCHEMBL15401046 0.91 GSK3A (0.38) GSK3AGSK3BFLT3
SCHEMBL9977700 0.91 GSK3A (0.38) GSK3AGSK3BFLT3
SCHEMBL16199061 0.87 GSK3A (0.39) GSK3AGSK3BFLT3JAK2SRC
SCHEMBL15399800 0.87 GSK3A (0.39) GSK3AGSK3BFLT3JAK2SRC
SCHEMBL9977728 0.87 GSK3A (0.39) GSK3AGSK3BFLT3JAK2SRC
SCHEMBL16199028 0.85 AURKA (0.37) GSK3AGSK3BFLT3JAK2SRC
SCHEMBL15401369 0.83 CDK7 (0.38)
SCHEMBL9970812 0.83 CDK7 (0.38)
SCHEMBL15400687 0.83 GSK3A (0.42) GSK3AGSK3BFLT3JAK2SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8871774-B2 Inhibitors of influenza viruses replication VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-10-28 US disclosed