SCHEMBL16199066

SCHEMBL16199066

O=C(N[C@@H]1CCCC(Nc2nc(-c3n[nH]c4ncccc34)ncc2F)C1)N1CCCCC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 4/20 0.36
BTK Q06187 2/20 0.36
CDC7 O00311 1/20 0.36
DAPK3 O43293 1/20 0.36
ROCK2 O75116 1/20 0.36
PRKD3 O94806 1/20 0.36
MAP4K4 O95819 1/20 0.36
PAK4 O96013 1/20 0.36
PIM1 P11309 1/20 0.36
PRKACA P17612 1/20 0.36
CDK2 P24941 1/20 0.36
FLT3 P36888 1/20 0.36
CSNK1A1 P48729 1/20 0.36
CDK8 P49336 1/20 0.36
CLK2 P49760 1/20 0.36
GSK3B P49841 1/20 0.36
CDK7 P50613 1/20 0.36
CDK9 P50750 1/20 0.36
PRKX P51817 1/20 0.36
JAK3 P52333 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15399920 1.00 EGFR (0.36) EGFRBTKCDC7DAPK3ROCK2
SCHEMBL15400429 0.99 EGFR (0.37) EGFRBTKCDC7DAPK3ROCK2
SCHEMBL16199082 0.94 EGFR (0.38) EGFRBTKCDC7DAPK3ROCK2
SCHEMBL16199011 0.93 GBA1 (0.37) EGFRBTKCDC7DAPK3ROCK2
SCHEMBL16199405 0.93 BTK (0.37) EGFRBTKCDK2CDK9ALDH1A1
SCHEMBL16199053 0.91 EGFR (0.37) EGFRBTK
SCHEMBL15400583 0.91 EGFR (0.37) EGFRBTK
SCHEMBL16199085 0.91 EGFR (0.37) EGFRBTK
SCHEMBL15400115 0.91 EGFR (0.37) EGFRBTK
SCHEMBL15400112 0.91 EGFR (0.37) EGFRBTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8871774-B2 Inhibitors of influenza viruses replication VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-10-28 US disclosed