SCHEMBL16199752

SCHEMBL16199752

CCn1nc(C)c(C2=Cc3cc(CI)ccc3-c3c(C4CCCCC4)c4ccc(C(=O)NS(=O)(=O)C(C)C)cc4n3C2)c1C(=O)N1CCN(C)CC1

nearest known ligand 0.42

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 8/20 0.42
KCNH2 Q12809 6/20 0.40
SCN9A Q15858 6/20 0.36
CYP3A4 P08684 2/20 0.33
SCN5A Q14524 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL863034 0.91 KCNH2 (0.49) NR1I2KCNH2SCN9ACYP3A4SCN5A
SCHEMBL862723 0.85 NR1I2 (0.49) NR1I2KCNH2SCN9ACYP3A4SCN5A
SCHEMBL863082 0.84 KCNH2 (0.49) NR1I2KCNH2SCN9ACYP3A4SCN5A
SCHEMBL862819 0.82 KCNH2 (0.47) NR1I2KCNH2SCN9ACYP3A4SCN5A
SCHEMBL863159 0.82 KCNH2 (0.49) NR1I2KCNH2SCN9ACYP3A4SCN5A
SCHEMBL863009 0.82 KCNH2 (0.49) NR1I2KCNH2SCN9ACYP3A4SCN5A
SCHEMBL862641 0.79 KCNH2 (0.50) NR1I2KCNH2SCN9ACYP3A4SCN5A
SCHEMBL862991 0.78 KCNH2 (0.51) NR1I2KCNH2SCN9ACYP3A4SCN5A
SCHEMBL862678 0.78 KCNH2 (0.51) NR1I2KCNH2SCN9ACYP3A4SCN5A
SCHEMBL862925 0.77 NR1I2 (0.49) NR1I2KCNH2SCN9ACYP3A4SCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2396329-B1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL MYERS SQUIBB CO (US) 2014-10-29 EP disclosed