SCHEMBL16200020

SCHEMBL16200020

CC(Cc1ccc(-c2ccnc(NC3CC(C)(C)NC(C)(C)C3)n2)cc1)N=N

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 9/20 0.43
CDK1 P06493 5/20 0.38
CDK4 P11802 5/20 0.38
CCNA2 P20248 5/20 0.38
CDK2 P24941 5/20 0.38
CCNB1 P14635 4/20 0.38
CCND1 P24385 4/20 0.38
CCNA1 P78396 4/20 0.38
MAPK8 P45983 2/20 0.37
CCNE1 P24864 2/20 0.37
CCND3 P30281 2/20 0.37
CDK6 Q00534 2/20 0.37
ROCK2 O75116 3/20 0.35
KCNH2 Q12809 1/20 0.35
KDM4E B2RXH2 1/20 0.35
LMNA P02545 1/20 0.35
GAA P10253 1/20 0.35
MAPK9 P45984 1/20 0.35
MAPK10 P53779 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13633638 0.87 IKBKB (0.43) IKBKBCDK1CDK4CCNA2CDK2
SCHEMBL3477899 0.87 IKBKB (0.45) IKBKBCDK1CDK4CCNA2CDK2
SCHEMBL4489766 0.87 IKBKB (0.45) IKBKBCDK1CDK4CCNA2CDK2
SCHEMBL3472713 0.81 IKBKB (0.41) IKBKBCDK1CDK4CCNA2CDK2
SCHEMBL3477574 0.81 IKBKB (0.41) IKBKBCDK1CDK4CCNA2CDK2
SCHEMBL3478250 0.80 IKBKB (0.45) IKBKBMAPK8ROCK2KCNH2KDM4E
SCHEMBL13633601 0.80 IKBKB (0.39) IKBKBCDK1CDK4CCNA2CDK2
SCHEMBL3471613 0.79 IKBKB (0.49) IKBKBCDK1CDK4CCNA2CDK2
SCHEMBL4477031 0.79 IKBKB (0.40) IKBKBCDK1CDK4CCNA2CDK2
SCHEMBL4482129 0.79 SYK (0.46) IKBKBMAPK8ROCK2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1615898-B1 2-Aminopyrimidine derivatives and their medical use NOVARTIS AG (CH) 2014-10-29 EP disclosed