SCHEMBL162089

SCHEMBL162089

COC(=O)c1ccc(C(=O)OC)c(OC(F)(F)C(F)(Br)OC(F)(F)C(F)(F)C(F)(F)F)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.44
KDM4E B2RXH2 11/20 0.43
ALDH1A1 P00352 7/20 0.43
MAPT P10636 4/20 0.43
HSD17B10 Q99714 4/20 0.43
HPGD P15428 4/20 0.43
ATM Q13315 2/20 0.43
GAA P10253 2/20 0.43
GLA P06280 1/20 0.43
CASP1 P29466 1/20 0.43
CASP7 P55210 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.39
PDK2 Q15119 4/20 0.38
CFTR P13569 1/20 0.36
PDK1 Q15118 2/20 0.36
PDK3 Q15120 2/20 0.36
PDK4 Q16654 2/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2448891 0.94 NOTUM (0.40) NOTUMKDM4EALDH1A1MAPTHSD17B10
SCHEMBL1439810 0.87 NOTUM (0.43) NOTUMKDM4EALDH1A1MAPTHSD17B10
SCHEMBL1440552 0.84 NOTUM (0.45) NOTUMKDM4EALDH1A1MAPTHSD17B10
SCHEMBL175762 0.82 NOTUM (0.40) NOTUMKDM4EALDH1A1MAPTHSD17B10
SCHEMBL158528 0.81 CA12 (0.36) NOTUMKDM4EALDH1A1HSD17B10HPGD
SCHEMBL1444213 0.79 NOTUM (0.43) NOTUMKDM4EALDH1A1MAPTHSD17B10
SCHEMBL175588 0.78 KDM4E (0.40) NOTUMKDM4EALDH1A1MAPTHSD17B10
SCHEMBL158941 0.76 KDM4E (0.32) KDM4EALDH1A1HSD17B10HPGDGAA
SCHEMBL160470 0.75
SCHEMBL1440190 0.73 NOTUM (0.37) NOTUMKDM4EALDH1A1MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 26 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2611855-A1 POLYARAMID FILMS COMPRISING FLUOROVINYLETHER FUNCTIONALIZED AROMATIC MOIETIES E.I. Du Pont De Nemours And Company (US) 2013-07-10 EP disclosed
US-8350099-B2 Fluorovinyl ether functionalized aromatic diesters, derivatives thereof, and process for the preparation thereof E I DU PONT DE NEMOURS AND COMPANY (US) 2013-01-08 US disclosed
US-8350099-B2 Fluorovinyl ether functionalized aromatic diesters, derivatives thereof, and process for the preparation thereof E I DU PONT DE NEMOURS AND COMPANY (US) 2013-01-08 US disclosed
US-8350099-B2 Fluorovinyl ether functionalized aromatic diesters, derivatives thereof, and process for the preparation thereof E I DU PONT DE NEMOURS AND COMPANY (US) 2013-01-08 US disclosed
US-8304513-B2 Polyesters comprising fluorovinylether functionalized aromatic moieties E I DU PONT DE NEMOURS AND COMPANY (US) 2012-11-06 US disclosed
US-8304513-B2 Polyesters comprising fluorovinylether functionalized aromatic moieties E I DU PONT DE NEMOURS AND COMPANY (US) 2012-11-06 US disclosed
US-8304513-B2 Polyesters comprising fluorovinylether functionalized aromatic moieties E I DU PONT DE NEMOURS AND COMPANY (US) 2012-11-06 US disclosed
EP-2473474-A2 FLUOROETHER FUNCTIONALIZED AROMATIC DIESTERS AND DERIVATIVES THEREOF E. I. du Pont de Nemours and Company (US) 2012-07-11 EP disclosed
EP-2473547-A2 POLYARAMID COMPRISING FLUOROVINYLETHER FUNCTIONALIZED AROMATIC MOIETIES E. I. du Pont de Nemours and Company (US) 2012-07-11 EP disclosed
EP-2473543-A2 POLYESTERS COMPRISING FLUOROVINYLETHER FUNCTIONALIZED AROMATIC MOIETIES E. I. du Pont de Nemours and Company (US) 2012-07-11 EP disclosed
US-20110218317-A1 POLYESTERS COMPRISING FLUOROVINYLETHER FUNCTIONALIZED AROMATIC MOIETIES E.I. DU PONT DE NEMOURS AND COMPANY (US) 2011-09-08 US disclosed
US-20110218317-A1 POLYESTERS COMPRISING FLUOROVINYLETHER FUNCTIONALIZED AROMATIC MOIETIES E.I. DU PONT DE NEMOURS AND COMPANY (US) 2011-09-08 US disclosed
US-20110218317-A1 POLYESTERS COMPRISING FLUOROVINYLETHER FUNCTIONALIZED AROMATIC MOIETIES E.I. DU PONT DE NEMOURS AND COMPANY (US) 2011-09-08 US disclosed
US-20110218319-A1 POLYARAMID FILMS COMPRISING FLUOROVINYLETHER FUNCTIONALIZED AROMATIC MOIETIES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2011-09-08 US disclosed
US-20110213118-A1 POLYARAMID COMPRISING FLUOROVINYLETHER FUNCTIONALIZED AROMATIC MOIETIES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2011-09-01 US disclosed
US-20110213118-A1 POLYARAMID COMPRISING FLUOROVINYLETHER FUNCTIONALIZED AROMATIC MOIETIES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2011-09-01 US disclosed
US-20110213118-A1 POLYARAMID COMPRISING FLUOROVINYLETHER FUNCTIONALIZED AROMATIC MOIETIES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2011-09-01 US disclosed
WO-2011028791-A2 POLYARAMID COMPRISING FLUOROVINYLETHER FUNCTIONALIZED AROMATIC MOIETIES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2011-03-10 WO disclosed
WO-2011028778-A2 POLYESTERS COMPRISING FLUOROVINYLETHER FUNCTIONALIZED AROMATIC MOIETIES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2011-03-10 WO disclosed
WO-2011028767-A2 FLUOROETHER FUNCTIONALIZED AROMATIC DIESTERS AND DERIVATIVES THEREOF E. I. DU PONT DE NEMOURS AND COMPANY (US) 2011-03-10 WO disclosed