Diethylamine

Diethylamine

SCHEMBL16239552

CCNCC.CS(=O)(=O)NC(=O)c1cc(Cl)c(COc2cnc(C3CC3)c(C3CC3)c2)cc1F

nearest known ligand 0.64

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

CCKAR

The experimentally established mechanism targets of Diethylamine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 20/20 0.64
SCN5A Q14524 2/20 0.59
SCN2B O60939 1/20 0.59
SCN1A P35498 1/20 0.59
SCN1B Q07699 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14892882 0.96 SCN9A (0.69) SCN9ASCN5ASCN2BSCN1ASCN1B
SCHEMBL16239622 0.89 SCN9A (0.76) SCN9ASCN5ASCN2BSCN1ASCN1B
Diethylamine SCHEMBL16239701 0.88 SCN9A (0.58) SCN9ASCN5ASCN2BSCN1ASCN1B
Diethylamine SCHEMBL16178014 0.84 SCN9A (0.68) SCN9ASCN5ASCN2BSCN1ASCN1B
SCHEMBL364874 0.83 SCN9A (0.62) SCN9ASCN5ASCN2BSCN1ASCN1B
SCHEMBL16174929 0.82 SCN9A (0.86) SCN9ASCN5ASCN2BSCN1ASCN1B
SCHEMBL15036783 0.79 SCN9A (0.73) SCN9ASCN5ASCN2BSCN1ASCN1B
SCHEMBL16239561 0.79 SCN9A (0.64) SCN9ASCN5ASCN2BSCN1ASCN1B
SCHEMBL16178222 0.78 SCN9A (1.00) SCN9ASCN5ASCN2BSCN1ASCN1B
SCHEMBL16239769 0.77 SCN9A (0.67) SCN9ASCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593431-B1 N-SULFONYLBENZAMIDES AS INHIBITORS OF VOLTAGE-GATED SODIUM CHANNELS PFIZER LTD (GB) 2014-11-19 EP disclosed