SCHEMBL16239608

SCHEMBL16239608

CS(=O)(=O)NC(=O)c1cc(F)c(COc2ccc(C(F)(F)F)nc2)cc1F

nearest known ligand 0.65

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 19/20 0.65
SCN5A Q14524 2/20 0.65
MRGPRX4 Q96LA9 1/20 0.43
SCN2B O60939 1/20 0.43
SCN1A P35498 1/20 0.43
SCN1B Q07699 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16239784 0.86 SCN9A (0.62) SCN9ASCN5A
SCHEMBL16239716 0.85 SCN9A (0.70) SCN9ASCN5A
SCHEMBL16175152 0.84 SCN9A (0.63) SCN9ASCN5ASCN2BSCN1ASCN1B
SCHEMBL16239609 0.83 SCN9A (0.70) SCN9ASCN5A
SCHEMBL16239963 0.83 SCN9A (0.70) SCN9ASCN5A
SCHEMBL16240191 0.82 SCN9A (0.76) SCN9ASCN5A
SCHEMBL16239860 0.82 SCN9A (0.68) SCN9ASCN5ASCN2BSCN1ASCN1B
SCHEMBL16239910 0.82 SCN9A (0.78) SCN9ASCN5A
SCHEMBL16239610 0.82 SCN9A (0.74) SCN9ASCN5A
SCHEMBL16240139 0.82 SCN9A (0.74) SCN9ASCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593431-B1 N-SULFONYLBENZAMIDES AS INHIBITORS OF VOLTAGE-GATED SODIUM CHANNELS PFIZER LTD (GB) 2014-11-19 EP disclosed