SCHEMBL16274752

SCHEMBL16274752

O=C(Nc1ccccc1)c1c(O)c2c(Nc3ccccc3)ncnc2n(OCc2ccccc2)c1=O

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
EGFR P00533 5/20 0.45
ERBB2 P04626 1/20 0.45
MAPT P10636 1/20 0.40
AURKB Q96GD4 4/20 0.39
AURKA O14965 2/20 0.39
RET P07949 4/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
HIF1A Q16665 1/20 0.39
SGMS2 Q8NHU3 1/20 0.38
MTOR P42345 1/20 0.38
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 2/20 0.37
KDR P35968 1/20 0.37
INCENP Q9NQS7 1/20 0.37
HPGD P15428 1/20 0.37
HTT P42858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16275096 0.82 MEN1 (0.43) EGFRAURKAMEN1KMT2ASGMS2
SCHEMBL16274771 0.81 MAPT (0.43) EGFRMAPTAURKBAURKARET
SCHEMBL3516729 0.79 HIF1A (0.50) EGFRMAPTMEN1KMT2AHIF1A
SCHEMBL16274789 0.79 EGFR (0.42) EGFRERBB2MAPTAURKBKDM4E
SCHEMBL16274831 0.77 MEN1 (0.46) MEN1KMT2AKDM4EALDH1A1HTT
SCHEMBL16274762 0.73 KDM4E (0.47) EGFRMAPTKMT2AKDM4EALDH1A1
SCHEMBL16274598 0.71 KDM4E (0.46) EGFRMAPTMEN1KMT2AKDM4E
SCHEMBL16274895 0.71 KDM4E (0.46) EGFRMAPTKMT2AKDM4EALDH1A1
SCHEMBL16274992 0.71 KDM4E (0.46) EGFRMAPTKMT2AKDM4EALDH1A1
SCHEMBL16274897 0.71 KDM4E (0.45) EGFRMAPTKDM4EALDH1A1KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2810944-A1 HETEROCYCLIC COMPOUND HAVING ANTI-HIV ACTIVITY Toyama Chemical Co., Ltd. (JP) 2014-12-10 EP disclosed